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2-[(4-chlorophenyl)methyl]-5-[4-(pyrrolidin-1-yl)piperidine-1-carbonyl]-1,3-benzoxazole
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-3-methylurea
(2H-1,3-benzodioxol-5-ylmethyl)({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl})(pyridin-3-ylmethyl)amine
1-(2-{[3-(cyclohexyloxy)-2-hydroxypropyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
7-[(2-fluorophenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-[(methylsulfanyl)methyl]furan-2-carboxamide
7-cyclobutaneamido-N-(2-methoxyethyl)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
4-{2-oxo-2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethyl}piperazin-2-one
4-[(1-acetylpiperidin-4-yl)oxy]-N-[(2-aminopyridin-3-yl)methyl]-3-methoxybenzamide
2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
methyl 4-{[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)carbamoyl}butanoate
methyl (1S,3S,3aR,6aS)-5-ethyl-3-(1-methyl-1H-imidazol-5-yl)-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-({5-[(3,4-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
3-(2,3-dihydro-1H-inden-2-yl)-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
5-({4-[(2S)-2,4,5,5-tetramethylpiperazine-1-carbonyl]-1,3-oxazol-2-yl}methoxy)isoquinoline
N-[2-(2-methoxy-5-{[4-(2-methylphenyl)piperazin-1-yl]methyl}phenoxy)ethyl]-2-(trifluoromethyl)benzene-1-sulfonamide
3,3-dimethyl-1-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}urea
1-{1-[(tert-butylcarbamoyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-(4-hydroxyphenyl)-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
6-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-3,4-dihydroquinazolin-4-one
1-(5-chloropyridine-2-carbonyl)-2-(4-methylpiperazine-1-carbonyl)piperazine
N-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
N-{3-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]phenyl}acetamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-methylpiperidine-2-carboxamide
1-cyclopentyl-N5-(2-methylpropyl)-4-oxo-N3,N3-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}thiomorpholine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)-N-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}propanamide
N-(2-methoxyethyl)-1,3-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-ethoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(4-methoxyphenyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}cyclopentane-1-carboxamide
1-cyclopentyl-4-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperazine
2-[1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazol-5-yl]-1,3-thiazole
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}furan-2-carboxamide
2-[2-(2-methyl-1,3-thiazole-4-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
7-({[(4-chlorophenyl)(phenyl)methyl]amino}methyl)-5-[2-(piperidin-1-yl)ethyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(pyrrolidin-1-yl)piperidine
N-cyclopropyl-3-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]sulfamoyl}benzamide
5-(2-ethoxyphenyl)-4-phenyl-1-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}-1H-imidazole
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
[1-ethyl-5-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(4-methylphenyl)methyl]piperidine
2-chloro-4-({3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)phenol
[(3-ethyl-1,2-oxazol-5-yl)methyl]({[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl})amine
6-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2,3-dihydropyridazin-3-one
N-[(2-chlorophenyl)methyl]-N-methyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
(2S)-2,6-diamino-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}hexanamide
2-[2-(dimethylamino)ethyl]-9-[2-(1H-pyrazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(adamantan-1-ylmethyl)-2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide