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3-(4-chlorobenzoyl)-1-cyclopentylpiperidine
N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-methylbenzamide
(1S,5R)-3-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[methyl(2-phenylethyl)amino]-2-[2-(oxolan-3-yl)ethyl]-2,3-dihydropyridazin-3-one
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
6-[4-(2,1,3-benzothiadiazol-4-ylmethyl)piperazin-1-yl]pyrazine-2-carboxamide
4-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)-2-(trifluoromethyl)morpholine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyridine-3-carboxamide
(2R)-2-(hydroxymethyl)-N-[4-methoxy-3-(2-methoxyacetamido)phenyl]pyrrolidine-1-carboxamide
5-amino-1-[2-(4-chlorophenyl)morpholin-4-yl]pentan-1-one
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carboxamide
1-(2-methoxyphenyl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
2-amino-6-cyclobutyl-4-{2-[2-(dimethylamino)ethoxy]phenyl}pyridine-3-carbonitrile
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-5-(oxolan-2-yl)thiophene-2-carboxamide
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)piperazine
5-(oxolan-2-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]thiophene-2-carboxamide
1-ethyl-N-(furan-2-ylmethyl)-5-[4-(2-methoxyphenyl)piperazin-1-yl]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxamide
4-[2-(4-chlorophenyl)propyl]-4H-1,2,4-triazole
1-(9H-purin-6-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-4-amine
5-[1-(3,4-difluorobenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
8-[4-(piperidin-1-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-4-yl)ethan-1-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-(3-methoxypropyl)piperidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-(dimethylamino)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]benzamide
1-phenyl-4-(2,5,7-trimethylquinoline-4-carbonyl)piperazin-2-one
2-(2-hydroxypropyl)-9-[2-(thiophen-2-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(2-acetylphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
2-{[(2-hydroxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}-5,8-dimethylquinolin-4-ol
[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl](methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
2-{methyl[1-(pyridin-3-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-(2-methoxyethyl)piperidine
1-[1-(2-phenylethyl)-5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
methyl 1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidine-2-carboxylate
N-({7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
(2E)-N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-3-(thiophen-2-yl)prop-2-enamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-cycloheptyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-yl}benzoic acid
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N-[4-(furan-2-yl)phenyl]-1-[2-(morpholin-4-yl)ethyl]piperidine-3-carboxamide
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(3R,4R)-4-amino-1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}piperidin-3-ol
8-(oxolane-3-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-fluorophenyl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}cyclopropane-1-carboxamide
2-{1-[(4-methylphenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol