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5-(1-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}pyrrolidin-2-yl)-N-methylthiophene-2-carboxamide
1-(8-chloroquinolin-5-yl)-3-ethyl-3-[(1-ethylpyrrolidin-3-yl)methyl]urea
2-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1-phenyl-1H-1,2,4-triazol-3-yl}acetamide
8-[3-(1H-indol-3-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-aminoethyl)-N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]quinazolin-4-amine
4-(4-chlorophenyl)-1-(4,4-difluoropiperidin-1-yl)butan-1-one
5-methyl-2-{1-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
6-methyl-2-{2-[2-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
2-(2,4-difluorophenoxy)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
2-[2-(1-{[3-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
[(4-fluoro-3-methoxyphenyl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
2-({4-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)-1H-1,3-benzodiazole
3-{2-[4-(3-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
2-(furan-2-yl)-5-{1-[2-(pyridin-3-yloxy)propyl]-1H-imidazol-2-yl}pyrimidine
5-(4-cyclopentylpiperazine-1-carbonyl)-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-{2-[4-(trifluoromethyl)phenyl]ethyl}acetamide
[(3-chlorophenyl)methyl](ethyl)(oxan-4-ylmethyl)amine
1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-methyl-9-(5-methyl-1H-1,3-benzodiazole-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
4-[(6-chloroquinolin-2-yl)methyl]-1λ6-thiomorpholine-1,1-dione
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethylpyrimidine-5-carboxamide
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(naphthalen-1-ylmethyl)acetamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-1-ene-1-carboxamide
2-[(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)methyl]phenol
1-[(2,4-difluorophenyl)methyl]-3-(3-fluoro-4-methoxybenzoyl)piperidine
3-(pyrrolidine-1-carbonyl)-2-(3,4,5-trimethoxyphenyl)pyridine
2-methoxy-1-{3-[3-(pyridin-3-yl)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
3-[3-(dimethylamino)propyl]-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[(3R,5S)-1-[(2-fluorophenyl)methyl]-5-(morpholine-4-carbonyl)pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-[6-(propan-2-yl)pyridin-2-yl]piperazine
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
3-[(2R,3R,6R)-5-cyclopropanecarbonyl-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-4-methylpiperidine
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[butyl(4-hydroxybutyl)amino]-2-(5-fluoro-2-methoxyphenyl)acetic acid
2-(2-{[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
(4aS,8aR)-6-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-cyclopropyl-3-(2-{4-[(4-fluorophenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
(1S,5R)-3-methyl-N-(4-phenoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-{2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)morpholin-2-yl]ethyl}-2-hydroxyacetamide
N-[(3,4-dimethoxyphenyl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-(pyridin-3-ylmethyl)acetamide
2-(furan-2-yl)-1-(thiophene-3-carbonyl)azepane
1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
7-chloro-3-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
{2-[(4aS,7aR)-6,6-dioxo-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}urea
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-2-cyclopropylpyrimidine-5-carboxamide
4-({[(2-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]amino}methyl)hepta-1,6-dien-4-ol
N-[(3R,4S)-4-cyclopropyl-1-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]pyrrolidin-3-yl]acetamide