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4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(2-methylbutyl)pyrimidine
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylsulfanyl)acetamide
2-[2-(1H-pyrazol-1-yl)ethyl]-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
5-(1-methyl-1H-indol-2-yl)thiophene-2-sulfonamide
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
3-{2-[2-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
1-(pyrimidin-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
3-(2,5-dimethoxyphenyl)-1-(thiophene-3-carbonyl)pyrrolidine
9-[2-(morpholin-3-yl)acetyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})(quinolin-4-ylmethyl)amine
2,2-dimethyl-N-(3-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}pyridin-2-yl)propanamide
2-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N-(1H-indazol-5-yl)-3-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}benzamide
N-[2-(dimethylsulfamoyl)ethyl]-4-methylpyrimidine-5-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-[2-oxo-2-(3-propanoylpiperidin-1-yl)ethyl]-3-phenylpyrrolidine-2,5-dione
5-(2-chlorophenyl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}furan-2-carboxamide
N-cyclopropyl-5-[2-(4-fluorophenyl)-2-hydroxyacetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
5-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(2S,4R)-4-amino-N,N-diethyl-1-(5-fluoro-1,3-dimethyl-1H-indole-2-carbonyl)pyrrolidine-2-carboxamide
2,4,6-trimethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
(1R,5R)-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]pyridine-3-carboxamide
5-tert-butyl-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1,3,4-oxadiazol-2-amine
3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(naphthalen-1-yl)ethyl]propanamide
2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1-(morpholin-4-yl)ethan-1-one
N-methyl-2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]aniline
1-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}cyclopropane-1-carboxamide
(1R,3S)-7-{[3-(2-hydroxyethoxy)phenyl]methyl}-3-methoxy-7-azaspiro[3.5]nonan-1-ol
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-[4-(oxolan-2-yl)butyl]urea
ethyl 1-[(1S)-1-carbamoyl-2-methylpropyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
(4aS,7aR)-1-[4-(hydroxymethyl)benzoyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[4-({4-[3-(dimethylamino)-2-hydroxypropoxy]phenyl}methyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
5-[4-(butylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
4-(5-methoxyfuran-2-carbonyl)-2-(4-methylpentyl)morpholine
4-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-5-ethylfuran-2-carboxamide
4-(2-{1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-2-yl}ethyl)phenol
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
2-amino-6-(2-methylpropyl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]pyrimidine-4-carboxamide
4-(2,3-dihydro-1H-inden-2-yl)-11-[(3-methylbutyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-methyl-N-(2-phenoxyethyl)-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
4-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
N-[(3R,4S)-4-(propan-2-yl)-1-[2-(propan-2-yloxy)acetyl]pyrrolidin-3-yl]methanesulfonamide
2-(dimethylamino)-N-(2-methanesulfonylethyl)-2-(4-methylphenyl)acetamide
1-{[1-(quinoxalin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-({4-[3-(2-methylphenoxy)azetidine-1-carbonyl]phenyl}methyl)piperidine
2-[4-(6-aminopyrimidin-4-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
3-methyl-8-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(methylamino)-N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)pyridine-3-carboxamide
1-(2,4,6-trimethyl-3-{1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}phenyl)ethan-1-one