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ethyl 4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine-1-carboxylate
N,N-diethyl-2-({4-[2-(1H-imidazol-2-yl)benzoyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)acetamide
2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(1,2-oxazol-3-ylmethyl)acetamide
N-[3-(1H-imidazol-1-yl)propyl]-4-methyl-2-phenylpyrimidine-5-carboxamide
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-(1,2-oxazolidin-2-yl)propanamide
(5S,9aS,9bS)-5-(3-methoxyphenyl)-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[1-(4-chlorophenyl)cyclopropanecarbonyl]-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepan-5-one
1-[1'-(3-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
4-[4-(3,4,5-trimethoxyphenyl)phenyl]piperidin-4-ol
1-(5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
2-methyl-4-{3-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3-methylphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-methyl-5-(quinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-(methylamino)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}[2-(diethylamino)ethyl]ethylamine
4-{5-[1-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(ethoxymethyl)-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
4-[5-(2,3-difluoro-4-methoxybenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]-1H-pyrazole
(2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}ethyl)urea
2-(dimethylamino)-7-[3-(1H-pyrazol-4-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(3-methoxyphenyl)-1-[1-(3-phenylbutyl)piperidin-4-yl]ethyl]-N-methylpyridine-2-carboxamide
2-({4-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyridine
2-[1-(4-chloro-2-methylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]pyrazine
2-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[2-(dimethylamino)ethyl]-5-[1-(1H-indole-2-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
1-{2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
2-[(3-methoxyphenyl)methyl]-8-(oxan-4-yl)-2,8-diazaspiro[4.5]decan-3-one
(2R,6R)-4-(3-hydroxy-4-methylbenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(1-ethyl-2-methyl-1H-indol-5-yl)-3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
3-{2,7-diazaspiro[4.5]decane-2-carbonyl}-1,6-dimethyl-1,4-dihydroquinolin-4-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidine
3-({1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidin-3-yl}methyl)benzoic acid
5-(azepane-1-carbonyl)-N-cyclooctyl-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-5-(3-methoxyphenyl)-N-methyl-1,2,4-triazin-3-amine
4-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}morpholine
3-{[1-(3-cyclopentylpropyl)piperidin-4-yl]oxy}-N-cyclopropyl-4-methoxybenzamide
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-cyclopropylpropanamide
6-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(5S,9aS,9bS)-5-(4-methoxyphenyl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
2-methoxy-3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyridine
5-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-5-ethyl-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
7-chloro-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-N-(oxolan-2-ylmethyl)quinazolin-4-amine
4-(methoxymethyl)-5-methyl-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-1,2-oxazole-3-carboxamide
1-[3-(cyclopentyloxy)phenyl]-3-[3-(morpholin-4-yl)propyl]urea
N-[(3S,4R)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(3aR,6aR)-N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
(3R,5S)-5-[1-(2,4-dimethylphenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]pyrrolidin-3-ol
(3R,4S)-3,4-dimethyl-1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-4-ol