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N-(1-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
(1S,5R)-3-(1-benzothiophene-5-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-ethoxyethyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
5-(1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1H-1,2,3-triazol-4-yl)pyrimidine
N-[3-(2-fluorophenyl)propyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
1-{1-[1-cyclohexyl-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
1-(morpholin-4-yl)-3-{1-[(4-phenylphenyl)methyl]piperidin-3-yl}propan-1-one
2-{2-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
6-[2-(methylsulfanyl)benzoyl]-N-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-cyclopentyl-3-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
8-(3,4-difluorobenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(1-benzoxepine-4-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
3-(5-{[butyl(furan-2-ylmethyl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}pyrimidine-5-carboxylic acid
3-(4-methyl-1,3-thiazol-5-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
(3S,4R)-1-[(3-methylpyridin-4-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
N-[2-(2-methoxyphenyl)ethyl]-2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetamide
(1R,2R,4R)-N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
(2S,4R)-1-[(4-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N,N-dimethylpyrrolidine-2-carboxamide
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4-(furan-3-carbonyl)-1,4-diazepane
9-[2-(3-oxopiperazin-1-yl)acetyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)ethyl]-4-methylpiperazine
2-cyclopropyl-N-[2-(4-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]pyrimidine-5-carboxamide
4-{[5-(2H-1,3-benzodioxol-5-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]methyl}pyridine
5-methyl-1-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}-1H-pyrazole
2-(3-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
2-{3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]phenyl}-1H-1,3-benzodiazole
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1,2-oxazole-5-carboxamide
6-(aminomethyl)-N-[2-(2,3-dimethoxyphenyl)ethyl]-2-methylpyrimidin-4-amine
(1R,5R)-6-[2-(4-methoxyphenoxy)ethyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(3-methylphenyl)methyl]piperidin-3-yl}propanamide
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-3-(trifluoromethyl)benzene-1-sulfonamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2,4-difluorophenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
6-{[4-(2-hydroxyethoxy)phenyl]methyl}-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-{2-[cyclopentyl(methyl)amino]ethyl}-3-methyl-1-[3-(methylsulfanyl)phenyl]urea
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1-ethyl-2,5-dimethyl-1H-pyrrole-3-carboxamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]pentan-1-one
2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
1-benzyl-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-{3-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]phenyl}-1,3-thiazole
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2H-1,3-benzodioxole-5-carboxamide
4-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-4-yl}thiomorpholine
2-cyclopropyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1,3-benzoxazole-6-carboxamide
2-[(2R)-2-aminopropanoyl]-N-benzyl-N-methyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(carbamoylmethyl)piperidine-4-carboxamide
2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}benzonitrile
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(thiophen-3-yl)acetyl]pyrrolidine-3-carboxylic acid
2-(4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-1-yl)pyrazine