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2-(2-methoxyethyl)-6-(1,2-oxazolidine-2-carbonyl)-1,3-benzoxazole
5-ethyl-N-(1-ethyl-5-oxopyrrolidin-3-yl)thiophene-3-carboxamide
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]oxolane-3-carboxamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
1-(2-hydroxyethyl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(3-methoxypropyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
5-chloro-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
4-methyl-7-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-(1,3-benzothiazol-2-yl)-3-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]propanamide
N-[2-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)propyl]-2,2-diphenylacetamide
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(2-methylphenyl)piperidine
(cyclohex-3-en-1-ylmethyl)[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-5-(4,4,4-trifluorobutan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(2S)-1-hydroxy-4-methylpentan-2-yl]acetamide
4-(1-ethylpiperidin-4-yl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
8-(2,1,3-benzoxadiazol-4-ylmethyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 3-[(2E)-2-methylbut-2-en-1-yl]-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-(pyrrolidin-3-yl)benzamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
N-{1-[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclopropanecarboxamide
N-ethyl-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-(2-methylprop-2-en-1-yl)acetamide
N-({7-[(2E)-3-(2,6-difluorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1H-indole-5-carboxamide
2-[1-(4-chloro-2-methylphenyl)-5-(1-methoxypropyl)-1H-1,2,4-triazol-3-yl]acetamide
N-methyl-1-{[(2-methylnaphthalen-1-yl)carbamoyl]amino}cyclohexane-1-carboxamide
6-hydroxy-7-methoxy-4-[2-(3-methylphenyl)pyrimidin-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
(2S,4S)-4-amino-N-ethyl-1-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)pyrrolidine-2-carboxamide
2-benzyl-9-(5-propyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(3-methoxybenzoyl)piperazine
3-cyclopropyl-1-phenyl-5-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}-1H-1,2,4-triazole
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)-1H-pyrrole-2-carboxamide
N-(1-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
1-[3-(1H-imidazol-2-yl)benzoyl]-3-(2-methoxybenzoyl)piperidine
2-ethyl-5-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}pyrimidine
3-(5-acetylthiophene-3-carbonyl)-9-methoxy-N-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(9H-purin-6-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-hydroxy-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-[1-(1-{[2-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
4-(1H-1,2,3,4-tetrazol-1-ylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]benzamide
1-(1H-1,3-benzodiazol-2-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-({4-[(cyclopropylcarbamoyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}methyl)benzoic acid
N-(1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazin-2-one
2-[3-(benzyloxy)propyl]-5-(4-methylpiperazin-1-yl)-2,3-dihydropyridazin-3-one
7-(1,3-benzothiazol-2-yl)-4-(2-fluorobenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-methoxy-5-methylphenyl)-2-({5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}formamido)acetamide
N-benzyl-2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-ethylacetamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-phenylbutanamide