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(3E)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]hex-3-en-1-one
4-[2-(4-fluorophenoxy)ethyl]benzamide
N,N-dimethyl-2-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
N-[3-(3-methylphenyl)phenyl]-1-(thian-4-yl)piperidine-3-carboxamide
methyl 4-{[(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-2-[(2-methoxyethyl)carbamoyl]pyrrolidin-1-yl]methyl}benzoate
(2R,6R)-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3R,5S)-1-(2-methylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[3-(morpholin-4-yl)propyl]piperidine-3-carboxamide
(9aR)-8-(4-methoxybenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{2-[4-(2-cyclopentylethyl)-1H-1,2,3-triazol-1-yl]ethyl}(methyl)amine
5-cyclopropyl-N-ethyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
2-(quinolin-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
4-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-3-yl}-5-(4-fluorophenyl)-2-methylpyrimidine
3-({[(3,4-dimethoxyphenyl)methyl]amino}methyl)-N,N,7-trimethylquinolin-2-amine
1-(3-{[4-(1H-imidazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenyl)-3,5-dimethyl-1H-pyrazole
(2S)-2-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}-4-(methylsulfanyl)butan-1-ol
5-ethyl-2,3-dimethyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(6-chloro-3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)azocane
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(2-methoxybenzoyl)piperazine
N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]-1,2-oxazole-3-carboxamide
[(4-ethyl-5-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
ethyl(2-methylprop-2-en-1-yl){[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
N4-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-fluoro-N-methyl-N-{2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
3-[(4-methoxyphenyl)methyl]-1-methyl-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-(benzyloxy)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}butan-1-one
2-methyl-3-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine-1-carbonyl)-1,2,3,4-tetrahydroisoquinoline
1-(4-methoxybenzoyl)-4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazine
2-cyclopropyl-6-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-1,3-benzoxazole
5-cyano-N,4-dimethyl-6-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,6-dihydropyridine-3-carboxamide
N-(1-{7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
N-[4-(3-methoxyphenyl)phenyl]-1-(3-methoxypropanoyl)pyrrolidine-2-carboxamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(morpholin-4-yl)propanamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[(5-methylthiophen-2-yl)methyl]benzamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[(4-chlorophenyl)methyl]-3-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}urea
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(propan-2-yl)acetamide
2-(5-ethylpyridin-2-yl)-1-methyl-1H-1,3-benzodiazole
1-{4-[3-({[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
2-{1-[(8-chloroquinolin-2-yl)methyl]piperidin-4-yl}-N-methylacetamide
(2R)-2-amino-3-(ethylsulfanyl)-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]propan-1-one
(2S)-2-[({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)amino]-4-methylpentanamide
3-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-methylpyridazine
1-{4-[4-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-ol
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-chloro-N-(propan-2-yl)-4-({[1-(pyrazin-2-yl)propan-2-yl]carbamoyl}amino)benzamide
1-[(3-methoxyphenyl)methyl]-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-(2-hydroxyethyl)-2-(2-methoxyphenyl)-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide