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2-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-N-ethylpyrimidin-4-amine
3-[2-(4-cyclohexyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-cyclopentyl-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
3-(2-amino-1,3-thiazol-4-yl)-1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1-(5-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}thiophen-2-yl)ethan-1-one
methyl 5-[(adamantan-2-yl)amino]-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-({[1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
5-benzyl-5-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propylsulfanyl)ethan-1-one
1-(piperidin-3-ylmethyl)-4-(pyridin-3-yl)piperazine
6-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
3-benzyl-8-(oxan-4-yl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclopentanecarbonyl-N-[1-(pyrazin-2-yl)propan-2-yl]piperidine-4-carboxamide
[(2S,6S)-4-(6-methylpyridine-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
1-(cyclohexylmethyl)-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-2-one
N-({3-methyl-7-[(4-methyl-1H-imidazol-5-yl)methyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
4-[(4-methoxyphenyl)methyl]-1-[3-(trifluoromethyl)benzoyl]-1,4-diazepan-5-one
1-{1-[(3,5-difluorophenyl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
2-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-6-methylphenol
N-methyl-3-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridin-2-amine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
methyl 1-(2-methyl-6-propylpyrimidin-4-yl)piperidine-4-carboxylate
2-methyl-7-(3-methylbenzenesulfonyl)-2,7-diazaspiro[4.5]decane
(2S,4R)-4-amino-N-ethyl-1-(naphthalene-2-sulfonyl)pyrrolidine-2-carboxamide
3-(naphthalene-2-carbonyl)-1-(propane-1-sulfonyl)piperidine
5-fluoro-2-(3-methyl-1H-1,2,4-triazol-5-yl)-1H-indole
2-[methyl(propan-2-yl)amino]-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}acetamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(propan-2-yl)-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
3-(2,3-dihydro-1H-inden-4-yl)-1-(furan-2-ylmethyl)-1-[2-(morpholin-4-yl)ethyl]urea
N-(1-carbamoylcyclopentyl)-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
2-{[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}benzonitrile
1-methyl-4-{[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(1,2-oxazol-3-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
5-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-1-propyl-1H-pyrazole-4-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(2-oxopyrrolidin-1-yl)butanamide
2-butyl-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-{[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]methyl}-4-methyl-2H-chromen-2-one
5-(methoxymethyl)-N-[(4-methoxyphenyl)methyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-(4-methylpiperazin-1-yl)propanamide
3-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}benzoic acid
2-methoxy-5-{[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
N,N-bis(prop-2-en-1-yl)-2-[4-(pyridin-4-yl)-1,4-diazepan-1-yl]acetamide
4-[4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperazine-1-carbonyl]morpholine
N-({5-[(5-methylthiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
3-({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)pyrazine-2-carbonitrile
1-(1,3-dihydro-2-benzofuran-5-yl)-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
5-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide