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14-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-cyclopropyl-2-{[1-(1,4-dithiepan-6-yl)piperidin-4-yl]oxy}-4-methoxybenzamide
4-({1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
3-[(3R,4S)-1-{2-[4-(hydroxymethyl)phenyl]acetyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-(3-methylphenyl)benzamide
methyl (2S,4S,5R)-5-(2-chlorophenyl)-4-(cyclopentylcarbamoyl)-1,2-dimethylpyrrolidine-2-carboxylate
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
4-[({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)amino]-1-phenylpyrrolidin-2-one
(2S,4S)-4-amino-N-ethyl-1-[(4-ethylpiperazin-1-yl)sulfonyl]pyrrolidine-2-carboxamide
11-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-[(3-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-fluoro-4-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine
ethyl 4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine-1-carboxylate
2-(6-aminopyridin-3-yl)-2-[4-(2-ethoxyphenyl)piperazin-1-yl]acetic acid
N-methyl-N-(2-methylpropyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-{3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
2-(dimethylamino)-2-(2-methylphenyl)-N-[3-(methylsulfanyl)propyl]acetamide
5-[(cyclopropylmethyl)amino]-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(8-{[4-(diethylamino)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-3-fluorobenzamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
4-{1-[6-(2,5-dihydro-1H-pyrrol-1-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
4-cyclopentyl-11-[(3-methylbutyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(dimethylamino)-8-(6-methylheptan-3-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
8-{[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}quinoline
1-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
7-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
1-(2,2-dimethyloxane-4-carbonyl)-4-(3-methoxybenzoyl)piperazine
N-(3-{[(4-fluorophenyl)methyl]sulfanyl}propyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N,4-dimethyl-5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
7-[(2,4-dimethoxyphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-{3-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-pyrazol-5-yl)acetamide
4-[4-(2,2-dimethylpropyl)piperazin-1-yl]-2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(5-{1-[2-(morpholin-4-yl)ethyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
4-{3-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl]phenyl}-2-methylbutan-2-ol
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[(4-fluorophenyl)methyl]-1,4-diazepane
1-[(2-chlorophenyl)methyl]-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
1-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)propan-1-ol
2-{4-[1-(2-fluorophenyl)piperidin-4-yl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(5-phenyl-1,2,4-triazin-3-yl)azocane
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(2E)-2-methylbut-2-en-1-yl](oxolan-2-ylmethyl)amine
2-(2,5-dimethoxybenzenesulfonyl)-8-methyl-2,8-diazaspiro[4.5]decane
N,1-dimethyl-N-(2-methylpropyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{1-[(6-chloro-2H-chromen-3-yl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
methyl 3-(2-methoxyacetamido)-1-(3-phenylpropyl)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S,4R)-4-amino-N,N-diethyl-1-(pyridazine-3-carbonyl)pyrrolidine-2-carboxamide