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1-{4-[2-(3,4-dimethoxyphenyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-methylpropan-1-one
9-(2-methoxyethyl)-1-methyl-10-oxo-N-phenyl-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
5-[1-(naphthalene-1-carbonyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
1-(2,6-dichlorophenyl)-3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
1-(4-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}thiophen-2-yl)ethan-1-one
N-methyl-N-(1-methylpiperidin-4-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(2R,3R)-2-ethoxy-1'-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
(3aS,6aR)-5-[6-(dimethylamino)pyrimidin-4-yl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
2-(2-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)-N-methyl-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]acetamide
methyl 1-(2-methoxyethyl)-5-{[(2-methoxyphenyl)methyl]amino}-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,5R)-3-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(1,3-benzothiazol-6-yl)-1-[(4-phenyloxan-4-yl)methyl]urea
N-[(3R,4R)-3-hydroxy-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl]pyridine-2-carboxamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)butan-1-one
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(pyridin-2-ylmethyl)acetamide
2-(3-phenylpyrrolidin-1-yl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]ethan-1-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-1-ethyl-1H-pyrazole-4-carboxamide
5-{[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-ethylpyrimidin-2-amine
5-(isoquinolin-5-yl)-2-methoxybenzamide
9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
methyl 3-[1-(2-phenylethyl)-3-[(pyridin-2-ylmethyl)carbamoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoate
4-methyl-2-(1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
2,5,6-trimethyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
(1S,5R)-3-cyclobutanecarbonyl-6-(5-methoxyfuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}pyridine
N-({7-[4-(furan-2-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
[4-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenyl]methanol
N-[(5-chloro-1H-indol-2-yl)methyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
3-(2-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-5,5-dimethyl-1,3-oxazolidine-2,4-dione
N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-ethyl-7,8-dimethyl-N-(propan-2-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-4-sulfamoylbenzamide
(2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-(4-methyl-1,4-diazepane-1-carbonyl)pyrrolidine-2-carboxylic acid
2-cyclohexyl-N-methyl-N-(oxan-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
3-(2-methoxyphenyl)-1-methyl-3-{2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(methylsulfanyl)propan-1-one
N-(pyridin-3-ylmethyl)-4-[4-({[3-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]benzamide
1-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carboxamide
1-{1-[6-(3-chlorophenyl)-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridine-3-carbonyl]piperidin-4-yl}piperidin-4-ol
N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-oxo-2H-chromene-3-carboxamide
N-cyclopropyl-N-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)furan-2-carboxamide
2-[4-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-3,5-dimethyl-1H-pyrazol-1-yl]ethan-1-ol
2-{2-[2-(3,5-dichloropyridin-4-yl)-1H-imidazol-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-{1-[5-(hydroxymethyl)furan-2-carbonyl]piperidin-3-yl}-3-phenylpropan-1-one
3-[(4-fluorophenyl)methyl]-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-1,2-oxazole-5-carboxamide