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N-[3-(1H-imidazol-1-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
5-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N-(2-{3-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]phenoxy}propyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-methyl-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-indole
N-[1-(1-{[3-(difluoromethoxy)phenyl]methyl}-1,2,3,6-tetrahydropyridin-4-yl)ethyl]-N-methylacetamide
3-(2-{2-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-5-methyl-1,2,4-oxadiazole
2-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-3-yl]-1H-1,3-benzodiazole
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]acetamide
N-benzyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
dimethyl({4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}methyl)amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyridine-3-carboxamide
N-[3-(3-ethylphenoxy)propyl]-2-methoxy-N-methylpyrimidine-5-carboxamide
N,N-dimethyl-6-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]cyclopentanecarboxamide
1-({1-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
2-[4-(3-acetylphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
6-(3-fluorophenyl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{3-[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-oxopropyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(2H-1,3-benzodioxol-5-yloxy)ethan-1-one
3-ethyl-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
5-{3-[4-(2,4-dimethylphenyl)piperazin-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
6-{[4-(2-fluoro-4-methanesulfonylphenyl)piperazin-1-yl]methyl}-1,4-oxazepan-6-ol
3-(1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperidin-3-yl)-1-(4-methylpiperazin-1-yl)propan-1-one
2-{[2-(4-fluorophenyl)morpholin-4-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
3-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2,5-dimethyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-(1,3-benzothiazol-2-yl)-N-methyl-N-(pyrimidin-4-ylmethyl)propanamide
4-[3-(2-aminoethyl)phenyl]-N-cyclopentyl-1H-pyrrolo[2,3-b]pyridin-6-amine
5-(2-cyclopentylacetamido)-N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
1-(4-{[1-(1H-pyrazol-1-yl)propan-2-yl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-methyl-3-phenyl-8-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,8-diazaspiro[4.5]decane
(1S,5R)-6-(oxane-4-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(1,3-thiazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyrazin-2-amine
2,3-dimethyl-6-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-(2-ethylpiperidin-1-yl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
3,5-dimethyl-2-[({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}amino)methyl]pyridin-4-ol
5-(2-ethoxyphenyl)-4-(4-methylphenyl)-2-(4-methylpiperazin-1-yl)pyrimidine
4-[(2,3-dimethoxyphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
3-(3-acetylphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
3-(5-chloro-2-methoxybenzoyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
1-[4-fluoro-3-(2-methylpropanamido)phenyl]-5-oxopyrrolidine-3-carboxylic acid