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[(4-ethylphenyl)methyl](methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[4-(1-benzofuran-2-ylmethyl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
methyl({[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(2-phenylethyl)amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-amine
methyl 4-{[methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}benzoate
5-cyclopropanecarbonyl-1'-(3-methyl-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(propan-2-yl)-6-[4-(propan-2-yl)piperazin-1-yl]pyrimidin-4-amine
1-ethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]-4-phenylpiperazine
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-(4-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenoxy)pyrimidine
{3-[(2-methylphenyl)methyl]-1-(quinoxalin-2-yl)piperidin-3-yl}methanol
N-(adamantan-1-yl)-2-oxo-6-[(4-phenylpiperidin-1-yl)methyl]-1,2-dihydropyridine-3-carboxamide
({1-[1-(2-cycloheptylacetyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)urea
[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methanol
4-{3-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]pyridin-2-yl}morpholine
N-[2-(dimethylamino)ethyl]-3-{1-[1-(2-fluorophenyl)piperidin-4-yl]piperidin-4-yl}propanamide
1-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-(pyridin-3-yl)piperidin-4-ol
N-(isoquinolin-5-ylmethyl)-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
N-cyclopentyl-4-{4-[methyl(quinoxalin-6-ylmethyl)amino]piperidin-1-yl}benzamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2,2-dimethyl-N-[1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide
5-(2-methoxyphenoxymethyl)-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-cyclobutanecarbonyl-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane
3-tert-butyl-1-{4-[4-(piperidine-1-carbonyl)phenyl]phenyl}urea
3-(oxolan-3-yl)-5-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1,2,4-oxadiazole
N-(3-chloro-4-methoxyphenyl)-3-[1-(thian-4-yl)piperidin-3-yl]propanamide
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-[3-(propan-2-yloxy)propyl]propanamide
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
3-{[1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidin-3-yl]methyl}benzamide
5-{[3-(3-chlorophenyl)pyrrolidin-1-yl]methyl}-1-methyl-1H-imidazole
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl})amine
(1S,9S)-11-[6-(aminomethyl)-2-methylpyrimidin-4-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)urea
4-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-propylpyrrolidin-2-one
9-[(2R)-2-methoxy-2-phenylacetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(oxan-3-ylmethyl)-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-5-methylthiophene-2-carboxamide
6-[(diethylamino)methyl]-N-[1-(hydroxymethyl)cyclopentyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(2-methoxyethyl)-8-(1-methoxypropan-2-yl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(1H-indol-3-yl)-1-{4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
N-(2,2-dimethyloxan-4-yl)-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}propan-1-one
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1-methylazepane-2-carboxamide
6-(benzyloxy)-4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
1-cyclopentyl-N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
ethyl 4-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)piperazine-1-carboxylate
N-{3-[2-(1-phenylethyl)-1H-imidazol-1-yl]phenyl}methanesulfonamide
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide