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methyl (2S,4R)-1-[(3-ethoxy-4-hydroxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
1-cyclopropanecarbonyl-N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
N,1-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(4-fluoro-3-methoxyphenyl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
N-(1,3-benzothiazol-2-ylmethyl)-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-(3-chloro-2-propoxyphenyl)-3-methyl-3-(oxolan-3-ylmethyl)urea
2-methoxy-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenylacetamide
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-[3-(1H-pyrazol-1-yl)propyl]pyrimidine-5-carboxamide
methyl 3-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
1-{3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
5-acetamido-1-(2-methoxyethyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
3-cyclobutyl-4-[2-(propan-2-yl)pyrimidin-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butanamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]methylamine
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]acetamide
N,N,7-trimethyl-2-(1-{[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-1H-pyrazol-4-yl)quinoline-4-carboxamide
1-cyclobutanecarbonyl-N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]piperidine-4-carboxamide
N-({1-[(2E)-3-(1H-imidazol-4-yl)prop-2-enoyl]piperidin-3-yl}methyl)furan-2-carboxamide
N-{[1-(2,3-dihydro-1H-inden-4-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}methanesulfonamide
N-(1-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
2-(2,3-difluorophenoxymethyl)-N-[(4-ethylphenyl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
7-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
8-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(furan-2-carbonyl)-N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1,4-diazepane-1-carboxamide
5-{4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indole
2-(adamantan-1-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
2-[1-(1-methylpiperidin-4-yl)-4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperazin-2-yl]ethan-1-ol
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-(1-phenylcyclopropyl)acetamide
1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-3-(2-ethoxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-(2-methoxyethyl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(propan-2-yl)propanamide
1-(3-methylpiperidin-1-yl)-3-[(prop-2-en-1-yl)(prop-2-yn-1-yl)amino]propan-1-one
4-phenoxy-1-[3-(thiophen-3-yl)propanoyl]piperidine-4-carboxylic acid
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(4-phenylpiperidin-1-yl)acetamide
9-{5-amino-[1,2,4]triazolo[4,3-c]pyrimidin-7-yl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-propyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1,3-thiazole-4-carboxamide
3-(3-phenylpropyl)-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
2-{5-[5-(2-chlorophenyl)furan-2-yl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
methyl 3-{[(2E)-3-(4-methoxyphenyl)prop-2-enamido]methyl}-5-[2-(1,3-thiazol-4-yl)acetamido]benzoate
1-(2-aminoethyl)-N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-(4-{2-[benzyl(methyl)carbamoyl]ethyl}piperidine-1-carbonyl)pyridin-1-ium-1-olate
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-{4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
N-[4-(3-fluorophenyl)phenyl]-1-(3,3,3-trifluoropropanoyl)piperidine-3-carboxamide
N-[(2R,3R)-2-ethoxy-1'-[(3-hydroxy-4-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
2-(phenylamino)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide