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N-({1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
1-methyl-5-[({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]pyrrolidin-2-one
(2R,3R,6R)-5-(2-fluorobenzoyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-({4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}methyl)-1,4-oxazepan-6-ol
5-fluoro-2-{1-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
2-(2H-1,3-benzodioxol-5-yl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]acetamide
2-{9-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
N-(cyclopropylmethyl)-2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-4-(4H-1,2,4-triazol-4-yl)benzamide
2-ethyl-8-[4-(1H-pyrazol-3-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(methyl)[(5-methylthiophen-2-yl)methyl]amine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
1-(2-aminoethyl)-N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-{[(1R,5R)-3-(dimethylcarbamoyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
{5-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]furan-2-yl}methanol
4-(1H-indol-5-ylmethyl)-1-(3-methoxyphenyl)piperazin-2-one
5-chloro-4,6-dimethyl-3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
ethyl 1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
N6-(2,2-dimethyloxan-4-yl)-N5,N5-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-benzyl-N-ethyl-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
(3S)-N-tert-butyl-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-(1-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)pyrimidin-2-amine
(3R,4R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
benzyl({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})[(4-methyl-1,3-thiazol-5-yl)methyl]amine
[1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-2-yl]methanol
4-(furan-2-yl)-N-{[8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
N-(2-methoxyethyl)-N-methyl-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
7-(1,3-benzothiazol-2-yl)-4-[(4-methylphenyl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-3-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(thiomorpholin-4-yl)ethan-1-one
N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
4-fluoro-N-({1-[2-(2-methylphenyl)acetyl]piperidin-3-yl}methyl)benzamide
(3R,4R)-4-ethyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine-3,4-diol
1-[3-(1H-imidazol-1-yl)propyl]-4-(naphthalen-2-yl)-1H-1,2,3-triazole
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(oxan-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
ethyl 4-(2-{4-[2-(phenylsulfanyl)acetamido]-1H-pyrazol-1-yl}acetamido)piperidine-1-carboxylate
1-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]propanamide
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-3-[4-(methylsulfanyl)benzoyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[(3-fluorophenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
7-methyl-2-(thiophen-3-yl)-4-[(2,3,4-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-{6-[(propan-2-yl)amino]pyrimidin-4-yl}piperazin-1-yl)pyridine-3-carbonitrile
methyl 3-{[4-(4-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]sulfonyl}thiophene-2-carboxylate
2-(2-aminoethyl)-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(3-ethoxy-2-hydroxypropyl)benzamide
7-[(3,4-difluorophenyl)methyl]-2-(2-methylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-{4-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-ethylbutan-1-one
2-cyclopropyl-N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide