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N-{[8-(2-acetylbenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-(1,2-oxazinan-2-yl)propanamide
N-(2-phenoxyethyl)-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-ethyl-N-(2-methylprop-2-en-1-yl)-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-ethyl-1-methyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2,2-diphenyl-1-[7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
3-{[(2,3-dimethoxyphenyl)methyl]amino}-5-(dimethylsulfamoyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]benzamide
N-cyclohexyl-3-{[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]amino}propanamide
2-[(4-chlorophenyl)methyl]-8-[(2-fluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
6-[(4-fluorophenyl)methoxy]-4-[(4-hydroxyphenyl)methyl]-1-(propan-2-yl)-1,4-diazepan-2-one
1-[(5-carbamoyl-1,2,4-oxadiazol-3-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
5-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(pyrrolidine-1-carbonyl)pyridine
N-(4-{4-[(1,4-dioxan-2-ylmethyl)amino]piperidin-1-yl}phenyl)-2-phenoxyacetamide
1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
2-(3-chlorophenyl)-2-hydroxy-1-{4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-benzyl-1-{1,3-dioxo-2-[(3,4,5-trimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
2-{2,8-diazaspiro[4.5]decan-2-ylmethyl}-5-methylphenol
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(thiophen-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}pyridine-4-carboxamide
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
2-methyl-1-(5-{1H-pyrazolo[3,4-b]pyridin-1-yl}thiophen-2-yl)propan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethan-1-one
1-butyl-2-(4-methylpentanesulfonyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-imidazole
4-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
5-(4-acetylphenoxymethyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
1-(2-methoxyphenyl)-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(propan-2-yl)-1H-1,2,4-triazole
2-benzyl-9-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-({7-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
N-[(2R,3R)-1'-(2-ethylbutyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
1-(1-methanesulfonylpyrrolidine-2-carbonyl)-4-(2-methylphenoxy)piperidine
6-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyrimidin-4-amine
1-(oxolane-3-carbonyl)-3,3-diphenylpiperidine
(3S,4S)-1-[(3-fluoropyridin-4-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
4-benzyl-2-{[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
6-ethyl-2-oxo-N-[1-(phenylcarbamoyl)piperidin-4-yl]-1,2-dihydropyridine-4-carboxamide
5-{2-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({7-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
1,9-dimethyl-4-(2-propoxyethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl 2-[(3-fluorophenyl)sulfamoyl]-6-(3-methylbenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3R,4R)-3-methyl-1-(4-methylpyrimidine-5-carbonyl)-4-(oxan-4-yl)piperidin-4-ol
1-(3-methoxypropyl)-4-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-1,4-diazepan-6-ol
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1-benzothiophene-2-carboxamide
(3R,4S)-4-propyl-1-(5-propylpyrimidin-4-yl)pyrrolidin-3-amine
{[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}urea