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3-[2-(3-chlorophenyl)acetyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-3-ethylpiperazin-2-one
3-[(4-methoxyphenyl)methyl]-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-{1-[4-(1H-indol-3-yl)butanoyl]piperidin-4-yl}methanesulfonamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2,2,2-trifluoroethyl)acetamide
(2S,4R)-N-ethyl-1-methyl-4-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanamido}pyrrolidine-2-carboxamide
N-[2-(2-chloro-6-fluorobenzoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-2-methoxybenzamide
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-(thiolan-3-yl)pyridin-2-amine
N-{[8-(isoquinoline-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
3-methyl-4-oxo-N-[(4-sulfamoylphenyl)methyl]-3,4-dihydroquinazoline-7-carboxamide
2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-ol
1-phenyl-4-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]piperazin-2-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
methyl (2S,4R)-1-(2,2-diphenylethyl)-4-(4-fluorobenzamido)pyrrolidine-2-carboxylate
5-methyl-2-[5-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1H-1,3-benzodiazole
3-{benzyl[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-2-methylpropan-1-ol
1-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}azepan-2-one
4-[(2-cyanophenyl)methyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperazine-1-carboxamide
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-ethyl-1-[2-(1H-pyrazol-1-yl)ethyl]urea
[(4-fluorophenyl)methyl](1H-imidazol-2-ylmethyl)(pyridin-4-ylmethyl)amine
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
ethyl 4-[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidin-1-yl]piperidine-1-carboxylate
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(oxolan-3-yl)acetamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]propanamide
2-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,2,3,4-tetrahydroquinoline-6-sulfonamide
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(pyridin-4-ylmethyl)piperazine
(3aR,6aR)-2-benzyl-5-(cyclopentylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-1λ6-thiomorpholine-1,1-dione
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
2-[2-(dimethylamino)ethyl]-9-(3-fluoropyridin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-[5-(3-ethynylphenyl)-1,2,4-oxadiazol-3-yl]pyrimidine
N-{3-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-oxopropyl}acetamide
N,N-dimethyl-6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazin-2-amine
2-methoxy-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-phenylethan-1-one
5-tert-butyl-4-{[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}furan-2-carboxamide
3-(4-benzyl-1H-pyrazol-5-yl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
1-(5-chloropyridin-2-yl)-4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-[(2E)-3-phenylprop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
1-cyclopentyl-2-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
N-benzyl-N-methyl-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-4-yl}propanamide
8-chloro-2-(furan-2-yl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]quinoline-4-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(2-methyl-1H-indol-3-yl)acetamide
4-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}morpholine-2-carboxylic acid
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
[(5-chloro-2-methoxyphenyl)methyl](ethyl)[(4-methanesulfonylphenyl)methyl]amine
3-[(2,3-dimethoxyphenyl)methyl]-5-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione