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3-cyclohexyl-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
{3-benzyl-1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}methanol
ethyl 6-[4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxopiperazin-1-yl]pyridine-3-carboxylate
[1-(3-fluorophenyl)propan-2-yl][(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-cyclopropylacetamide
5-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]-1H-1,2,3-benzotriazole
7-[(3,5-dichloro-2-methoxyphenyl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-4-chlorophenol
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-amine
2-[4-(4-{[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-N-benzylacetamide
8-(2-methylpropyl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-fluorophenyl)-2-hydroxy-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
8-[3-methyl-4-(morpholin-4-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(3-methoxypropyl)-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
N-methyl-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(propan-2-yl)propanamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1-ethyl-6-oxopiperidine-3-carboxamide
2-{6-[1-(morpholin-4-yl)cyclohexanecarbonyl]-6-azaspiro[2.5]octane-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-methoxyphenoxy)ethan-1-one
N-(2-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]morpholin-2-yl}ethyl)acetamide
6-methoxy-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]pyrimidin-4-amine
2-ethyl-7-({3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}methyl)-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,N-dimethylazepan-4-amine
1-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]-3-methylbut-2-en-1-one
1-cyclopentyl-N3-(3-methylbutyl)-N5-[(1-methylpiperidin-3-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-{1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}ethan-1-ol
4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-2-amine
3-{1-[(2S)-2-acetamido-4-(methylsulfanyl)butanoyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
5-[4-(2-methylpyridin-4-yl)phenyl]-1H-imidazol-2-amine
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl](methyl)[(5-phenyl-1,2-oxazol-3-yl)methyl]amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-N-methyloxan-4-amine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
(3S,4R)-1-{[3-(2-hydroxyethoxy)phenyl]methyl}-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
4-({5-[2-(2-methoxyphenyl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
2-benzyl-N-[2-(dimethylsulfamoyl)ethyl]-1,3-thiazole-4-carboxamide
2,6-difluoro-N-(1H-imidazol-2-ylmethyl)-3-methylbenzamide
6-cyclopropyl-N-[3-(pyrrolidin-1-yl)propyl]pyrimidin-4-amine
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-[(4-phenoxyphenyl)methyl]pyrrolidin-3-ol
(1R,3S)-7-(2-amino-6-methoxypyrimidin-4-yl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
4-methyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
3-amino-1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
4-[4-({[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]but-3-yn-1-ol
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2,7-dimethylquinoline-4-carboxamide
1-(2-methoxyphenyl)-4-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
6-(morpholine-4-sulfonyl)-2-{spiro[2.3]hexane-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(4-methoxypyrimidin-2-yl)piperazin-2-yl}ethan-1-ol
N-[(3-methoxyphenyl)methyl]-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidin-4-amine
1-cyclopentyl-3-(2-fluorophenyl)-3-(2-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)pyrrolidine-2,5-dione