Tips: Press Ctrl key to select multiple functional groups
2-{[(3R,5S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]sulfanyl}-4-methylpyrimidine
N-ethyl-5-[8-methyl-4-(2-methylpyrrolidine-1-carbonyl)quinolin-2-yl]pyrimidin-2-amine
2-[4-(4-benzylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
N-[3-(benzyloxy)phenyl]-3-(hydroxymethyl)piperidine-1-carboxamide
2-{1-[(4-cyclopentylpyrimidin-2-yl)amino]ethyl}phenol
(3R,5S)-5-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]pyrrolidin-3-ol
3-(4-fluorophenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrazole-5-carboxamide
5-methyl-N-(3-{5-methyl-4-[(3-methyl-2-oxopentanamido)methyl]-1,3-oxazol-2-yl}phenyl)thiophene-2-carboxamide
N-{3-oxo-3-[2-(pyridin-2-yl)piperidin-1-yl]propyl}methanesulfonamide
N5-cyclopentyl-N6-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(quinoline-6-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
(2S,4S)-4-amino-1-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methylpyridine-2-carboxamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(1-phenylcyclopropyl)benzamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[(3S)-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl]acetamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(5-methylthiophene-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2,5-dimethoxyphenyl)-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-5-methyl-1,3-oxazole
1-[2-(methylamino)pyrimidine-5-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanamide
1-{[2-methyl-5-(trifluoromethyl)phenyl]methyl}piperidin-2-one
N-{[7-(4-acetylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
1-[2-(pyridin-2-yl)-4-{[2-(pyridin-2-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrrolidine-1-carboxamide
(3S,9aR)-3-(2-methylpropyl)-8-(naphthalene-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidine
1-[2-({[4-(butan-2-yloxy)-3-chlorophenyl]methyl}amino)ethyl]piperidin-4-ol
1-(3-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
9-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
2-{4-[(4-acetylpiperazin-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5,8-dimethyl-2-({[2-(oxan-2-yl)ethyl]amino}methyl)quinolin-4-ol
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(1H-indol-1-yl)ethan-1-one
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazole
1-[2-(4-chlorophenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-5-one
2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
5-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[3-(morpholin-4-yl)propyl]-3-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
3-{1-[(2S)-1-acetylpyrrolidine-2-carbonyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
(3S,7S,8aS)-7-{[(2-fluoro-5-methylphenyl)methyl]amino}-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
6-ethyl-1-methyl-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(pyrrolidin-1-yl)acetamide
N-(cyclobutylmethyl)-1-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-[4-(3-methoxyphenyl)piperazin-1-yl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propan-1-one
1-[4-methyl-2-({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)pyrimidin-5-yl]ethan-1-one
1-[(3S)-3-(dimethylamino)azepan-1-yl]-3-phenoxypropan-1-one
2-{4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazin-1-yl}-1,3-benzoxazole