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N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(dimethylamino)-2-(3-methylphenyl)acetamide
N-butyl-N-({1-[(4-cyanophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
3-[3,5-dimethyl-4-(pyrimidin-5-yl)-1H-pyrazol-1-yl]propanamide
6-oxo-1-(3-phenylpropyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}piperidine-3-carboxamide
5-chloro-2-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]phenol
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(pyridin-3-yl)acetamide
N-[2-(4-phenylpyrimidin-2-yl)ethyl]-4-(trifluoromethyl)pyrimidin-2-amine
3-(1H-imidazol-1-yl)-1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
(4aS,7aR)-1-[2-(1H-1,3-benzodiazol-2-ylmethoxy)acetyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2,2-diphenylethyl)-4-(1H-pyrrole-2-carbonyl)morpholine
10-methoxy-5-[1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
8-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
3-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-(2-methylpropyl)-1,2,4-oxadiazole
3-(benzylsulfamoyl)-5-(pyrimidin-5-yl)benzoic acid
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(1H-indol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1,1-dioxo-N-[4-(oxolan-2-ylmethoxy)phenyl]-1λ6-thiomorpholine-4-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-4-(pyridin-2-yl)pyrimidin-2-amine
4,4-difluoro-N-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)piperidine-1-carboxamide
2-ethyl-1-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine
N,N-diethyl-2-[(2-oxo-4-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}-1-(2-phenylethyl)-1,4-diazepan-6-yl)oxy]acetamide
4-[(2-hydroxyethyl)sulfamoyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)benzamide
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl][(3-phenyloxolan-3-yl)methyl]amine
N-[2-(4-fluorophenyl)ethyl]-2-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]acetamide
N-methyl-N-[(4-phenoxyphenyl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
2-[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-yl]-6-methyl-1H-1,3-benzodiazole
2-[1-(1-methanesulfonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1-(propan-2-yl)-1H-1,3-benzodiazole
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
4-(4-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
2-(4-chloro-2-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)acetic acid
6-fluoro-2-{2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}-1H-1,3-benzodiazole
1-(4,7-dimethylquinazolin-2-yl)-N-methyl-N-(propan-2-yl)piperidine-3-carboxamide
3-[2-chloro-5-(morpholin-4-yl)phenyl]-1-[(5-methylpyrazin-2-yl)methyl]urea
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2,5-dimethylfuran-3-carbonyl)piperidine-2-carboxamide
6-(5-chloro-2-fluorobenzoyl)-1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
1-cyclopentyl-3-(3-fluorophenyl)-3-{2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
1-[4-({[(5-ethylpyridin-2-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
7-(2,5-difluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-(4-methoxyphenyl)-3-methyl-4-{thieno[2,3-d]pyrimidin-4-yl}piperazin-2-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(3-methoxy-2-methylbenzoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-cyclopropyl-3-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-3-yl)propanamide
S-(4-fluoro-3-methylphenyl)-2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-oxoethane-1-sulfonamido
(2S)-2-[5-(5-ethylpyridin-2-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide