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2-(4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)quinazoline
5-{[(4-chlorophenyl)methyl]amino}-1-methyl-N-[2-(piperidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(4-{5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carbonyl}piperazin-1-yl)pyrimidine
N-[4-(3-methoxyphenyl)phenyl]-1-(oxane-4-carbonyl)pyrrolidine-2-carboxamide
8-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-methoxyethyl)-3-(1-methyl-1H-pyrazol-5-yl)-N-(naphthalen-1-ylmethyl)propanamide
(4aR,7aS)-4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-(2-methoxyphenyl)-4-[3-(3-methylpiperidin-1-yl)-3-oxopropyl]piperazin-2-one
1-(propan-2-yl)-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1H-pyrazole-4-carboxamide
1-(5-methyl-1,3,4-oxadiazol-2-yl)-4-(thian-4-yl)piperazine
4-(5-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
1-(3,5-dimethylphenyl)-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
5-{[3-(pyridin-2-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[1-(2-chlorophenyl)ethyl]-5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
2-(3-hydroxyphenyl)-N-[(6-methylquinolin-5-yl)methyl]acetamide
6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridin-3-amine
1-{[3-(5-methylfuran-2-yl)-1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyridin-2-one
6-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
N-[(4-fluorophenyl)methyl]-2-{2-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
(3R,9R)-11-[(4-phenyl-1,3-thiazol-2-yl)methyl]-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(pyridin-2-ylmethyl)piperidin-3-ol
1-(2-phenylethyl)-N-[(2-phenylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-(3-phenylpropyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-2-(pyrrolidin-1-ylmethyl)piperidine
3-fluoro-4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzene-1-sulfonamide
N-(3-cyano-4-methylphenyl)-4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazine-1-carboxamide
2-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}quinolin-8-ol
2-phenoxy-N-(1-{7-[(3,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
5-methanesulfonyl-1'-(3,3,3-trifluoro-2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-cyclohexyl-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-1-phenylcyclopropane-1-carboxamide
1,3-dimethyl-4-(5-phenoxyfuran-2-carbonyl)piperazin-2-one
1-[(3aS,6aS)-1-{[4-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[2,3-c]pyrrol-5-yl]-3-(1H-pyrazol-1-yl)propan-1-one
(4aS,7aR)-1-(2-chloro-4-fluorobenzenesulfonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(5-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2-(ethylamino)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]pyrimidine-5-carboxamide
(3aS,6aS)-2-acetyl-5-[benzyl(methyl)sulfamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-({cyclopropyl[(3-methylthiophen-2-yl)methyl]amino}methyl)pyridine-3-carboxylic acid
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
6-{[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]amino}-N,N-dimethylpyridine-3-carboxamide
methyl 6-[(piperidin-4-ylmethyl)amino]pyridine-3-carboxylate
4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
(1S,4S)-2-(3-chlorophenyl)-5-[(2S)-2-hydroxy-2-phenylacetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
5-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-methoxypyridine
1-ethyl-8-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-(1H-pyrazol-1-yl)acetamide
3-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}methyl)pyrrolidin-3-ol
4-methoxy-6-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyrimidin-2-amine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide