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(3S,4S)-1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
N-(1,3-dihydro-2-benzofuran-5-yl)-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
2-[1-(cyclohexylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-propyl-1,4-diazepan-5-one
N-(1-{1-[(6-fluoroquinolin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
2-(3-methylbutyl)-8-(3-methylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(4-fluorophenyl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(4-ethenylbenzoyl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-ethyl-1'-(5-methyl-1H-indazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]acetamide
4-(1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidine
(1,4-dioxan-2-ylmethyl)({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
2-(1-benzyl-1H-pyrazol-4-yl)-N,N,8-trimethylquinoline-4-carboxamide
N-(adamantan-1-yl)-2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(6-methoxynaphthalen-2-yl)ethyl]amine
5-tert-butyl-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,3,4-oxadiazol-2-amine
1-{4-[(2-benzylmorpholin-4-yl)methyl]thiophen-2-yl}ethan-1-one
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2,5-dimethoxybenzamide
1-(5-methyl-1,3-benzoxazol-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-ethyl-N-(pyridin-4-ylmethyl)-5-({[2-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(5,6-dimethylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-fluoro-4-methoxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
N-(5-fluoro-2-methylphenyl)-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-2,1,3-benzothiadiazole
ethyl 3-benzyl-1-(quinoline-8-sulfonyl)piperidine-3-carboxylate
3-(1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-2-yl)pyridine
N-(oxan-2-ylmethyl)-4-phenoxybutanamide
3-(2-methylpyrimidin-4-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
1-benzyl-4-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
N-benzyl-N,1-dimethyl-5-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2,2-dimethyloxane-4-carboxamide
1-[(4-{[1-(2-methoxybenzoyl)piperidin-3-yl]methoxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N,2-dimethyl-6-(piperidin-3-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-4-amine
3-(1H-pyrazol-3-yl)-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}piperidine-1-carboxamide
(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}piperidin-4-yl)methanol
N-methyl-3-(N-methyl-1-{2-phenylimidazo[1,2-a]pyridin-6-yl}formamido)butanamide
1-cyclopentyl-3-(3-fluorophenyl)-3-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
methyl 2-{3-oxo-1-[2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carbonyl]piperazin-2-yl}acetate
8-[(2S)-2-aminopropanoyl]-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(3,5-dichloro-4-methylbenzoyl)-1λ6-thiomorpholine-1,1-dione
N-benzyl-2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
N-[1-(4-hydroxyphenyl)propyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
5-(4-ethyl-2-methyl-1,3-thiazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-1-[3-(piperidin-1-ylmethyl)piperidin-1-yl]propan-1-one
(4S)-4-acetamido-5-oxo-5-(3-oxo-4-phenylpiperazin-1-yl)pentanamide
2-[4-(7-chloro-4-methylquinolin-2-yl)piperazin-1-yl]pyridine-3-carboxamide
N-{[(3S,4S)-1-[3-(furan-2-yl)benzoyl]-3-hydroxypiperidin-4-yl]methyl}propanamide