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ethyl 2-({3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carbonyl}amino)acetate
3-(pyridin-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[2-(1H-imidazol-1-yl)propyl]-2,3,6-trimethylquinoline-4-carboxamide
1-[(3-chloropyridin-4-yl)methyl]-4-(pyrrolidine-1-sulfonyl)piperazine
methyl 5-{[1-(4-fluorophenyl)propan-2-yl]amino}-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-(cyclopropylmethyl)-2-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
6-[(diethylamino)methyl]-N-[(1r,4r)-4-hydroxycyclohexyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(2S,4R)-N-ethyl-4-(5-methylthiophene-2-amido)-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
1-ethyl-8-[4-(4-methoxyphenyl)butan-2-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-(quinolin-4-yl)phenyl]acetamide
3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-[3-(morpholin-4-yl)propyl]propanamide
(4aR,8aS)-6-(4-methoxybenzoyl)-1-[2-(2-methoxyphenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-oxo-N-(pyrimidin-4-ylmethyl)-3,4-dihydroquinoxaline-2-carboxamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-[2-(pyridin-3-yl)acetyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrrolidine-3-carboxamide
{6-[4-(ethanesulfonyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}methanamine
4-[3-(azepane-1-carbonyl)piperidin-1-yl]-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-methoxy-5-({2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}methyl)benzoic acid
2,4-dichloro-3-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenol
N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)adamantan-1-amine
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
methyl 5-oxo-5-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)pentanoate
(3R,4R)-1-(1-ethyl-1H-indole-5-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
4-{[(2,3-dimethoxyphenyl)methyl]amino}-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-(1H-indol-4-ylmethyl)-4-(pyrrolidine-1-sulfonyl)benzamide
1-cyclopentyl-4-[5-(2,4-dimethylphenyl)-4-methyl-1H-imidazol-2-yl]pyrrolidin-2-one
(2S)-2-amino-1-[4-(benzenesulfonyl)piperazin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
1-{3-[4-(4-methylphenoxy)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
1-[(2-chlorophenyl)methyl]-N-[(3-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-methyl-5-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1,3-thiazole
6-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-N,N-dimethylpyrazin-2-amine
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-benzofuran-2-carboxamide
(2S,4R)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzoxazol-2-one
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-phenyl-N-[2-(pyridin-3-yloxy)propyl]-1H-pyrazole-4-carboxamide
methyl 4-(2-ethoxyphenyl)-1-methyl-1H-pyrrole-2-carboxylate
N-ethyl-N-[2-(3-methoxyphenoxy)ethyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
1-ethyl-2-{1-[2-(propan-2-yloxy)ethyl]-1H-1,2,3-triazol-4-yl}-1H-1,3-benzodiazole
1-(2-methylpropyl)-5-oxo-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}pyrrolidine-3-carboxamide
3-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[2-(morpholin-4-yl)ethyl]urea
N-[3-(4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}piperidin-1-yl)phenyl]pyridine-3-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(5-oxopyrrolidin-2-yl)acetamide
2-(6-methoxynaphthalen-2-yl)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]morpholine
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[3-(trifluoromethyl)phenyl]piperazine
3-(5-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
2-[1-(8-fluoroquinolin-2-yl)-N-[(2-methoxyphenyl)methyl]formamido]acetic acid
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(thiomorpholin-4-yl)pyridine-3-carboxamide