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2-[(benzyloxy)methyl]-4-(4-ethoxyphenyl)-1H-imidazole
(5S,9aS,9bS)-5-(3-ethoxy-4-methoxyphenyl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(9H-purin-6-yl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]piperidin-4-amine
2-[2-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[(3R,4R)-1-{6-[ethyl(methyl)amino]pyrimidin-4-yl}-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
N-butyl-1-cyclohexyl-5-[4-(4-methylphenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[2-(2-methyl-1H-indol-1-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(2-methoxyphenyl)-3-{2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[1-(thiophen-2-yl)ethyl]benzamide
2-(pyridin-2-yl)-7-{spiro[2.3]hexane-1-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
3-[(dipropylcarbamoyl)methyl]-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-(3-fluoro-4-methoxybenzoyl)-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
8-(1-benzofuran-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-chloro-3-ethyl-4-({8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1-methyl-1H-pyrazole
1-(4-{2,7-diazaspiro[4.5]decane-7-carbonyl}phenyl)imidazolidine-2,4-dione
5-acetamido-1-ethyl-N-(2-hydroxybutyl)-2-(3-methoxyphenyl)-1H-1,3-benzodiazole-7-carboxamide
N-[(1R,3S)-3-[(oxan-4-yl)carbamoyl]cyclopentyl]-1H-1,2,3-benzotriazole-5-carboxamide
N-[(2-fluorophenyl)methyl]-3-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}propanamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(1H-imidazol-2-yl)benzamide
4-(pyridin-3-yl)-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-ol
1-{2-[(2,2-dimethylpyrrolidin-1-yl)methyl]-5-methoxyphenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(2-methylphenoxy)ethan-1-one
3-{1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]pyrrolidin-3-yl]methanol
1-(2-fluorophenyl)-4-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]piperazine
5-(naphthalen-1-ylmethyl)-5-[3-oxo-3-(pyrrolidin-1-yl)propyl]pyrrolidin-2-one
3-benzyl-8-(cyclohexylmethyl)-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-2-amino-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-4-methylpentan-1-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(prop-2-ene-1-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-5-methoxy-3-methyl-1H-indole
2-(2,4-difluorophenyl)-5-(1,4-dithiepan-6-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-hydroxy-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-[(6-methylquinazolin-4-yl)amino]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-propyl-1,2-oxazole-3-carboxamide
1-ethyl-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}piperidine-2-carboxamide
N,5-dimethyl-N-[(5-methylthiophen-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
methyl (2R)-2-(4-hydroxyphenyl)-2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}acetate
5-(2,4-difluorophenoxymethyl)-N-[(3S)-2-oxoazepan-3-yl]-1,2-oxazole-3-carboxamide
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
N-[3-(4-{[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]amino}piperidin-1-yl)phenyl]-4-phenylbutanamide
5-{3-[2-(hydroxymethyl)piperidin-1-yl]-3-oxopropyl}-5-[(4-methoxynaphthalen-1-yl)methyl]pyrrolidin-2-one
N-(3,4-dimethoxyphenyl)-1-(oxan-4-yl)piperidin-3-amine
methyl 1-[9-methoxy-7-oxo-3-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]piperidine-2-carboxylate
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-cyano-5-fluorobenzamide
(1R,3s,6r,8S)-4-{3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-4-azatricyclo[4.3.1.13,8]undecane
3-(4-methoxyphenyl)-5-(2-propylpyrrolidine-1-carbonyl)-1H-pyrazole
1-(2-{4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-3,5-dimethyl-1H-1,2,4-triazole
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-6-oxopiperidine-3-carboxamide
1-(oxolane-2-carbonyl)-3,3-diphenylpiperidine