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1-(azocan-1-yl)-3-[2-methoxy-5-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
3-(3-hydroxy-3-methylbutyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
propan-2-yl (2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
2-{3-[(4-methyl-3-phenylpiperazin-1-yl)methyl]phenoxy}acetamide
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]propanamide
1-methyl-N-({8-[(3,4,5-trimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1H-pyrazole-3-carboxamide
2-[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-methyl-1-({3-[4-(pyrazin-2-yl)piperazine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}-1-[(3-methoxyphenyl)methyl]piperidine
5-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(3-phenylphenyl)piperidin-4-amine
methyl 4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]benzamide
1-{4-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
2-(4-ethylpiperazin-1-yl)-1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}ethan-1-one
3-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
2-(2-methoxyethyl)-6-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,3-benzoxazole
1-(3-cyanophenyl)-3-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}urea
1-ethyl-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-methyl-N-(pyrazin-2-ylmethyl)pyridin-2-amine
2-(2-fluorophenyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
3-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2-dihydroquinolin-2-one
4-[(benzyloxy)methyl]-1-[(3-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(1-{7-[(8-methoxyquinolin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
N-[(3R)-piperidin-3-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1-ethyl-N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}piperidine-2-carboxamide
2-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-2,3-dihydro-1H-isoindole
4-(3-hydroxy-3-methylbutyl)-N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]benzamide
2-[(2-fluorophenyl)methyl]-N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-1,3-benzoxazole-6-carboxamide
ethyl 1-(cyclopropylmethyl)-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[1-(3-chlorobenzoyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-[6-(3-methoxyphenoxy)pyridin-3-yl]urea
(4aS,7aR)-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(4-fluorophenyl)methyl]-5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-({5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)ethan-1-ol
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(5-methylpyrazin-2-yl)methyl]-1,2-oxazole-3-carboxamide
(4aR,7aS)-1-benzyl-4-(1-methyl-1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,3,6-trimethyl-N-(2-oxopiperidin-3-yl)quinoline-4-carboxamide
methyl 3-[(adamantan-1-ylformamido)methyl]-5-(furan-2-amido)benzoate
(2S,4R)-4-amino-1-[2-chloro-5-(piperidin-1-yl)benzoyl]-N-methylpyrrolidine-2-carboxamide
3-[5-(1-ethyl-2-oxo-1,2-dihydropyridin-4-yl)-3-methyl-1H-1,2,4-triazol-1-yl]-4-fluorobenzene-1-sulfonamide
6-(methoxymethyl)-N-[3-(morpholin-4-yl)propyl]pyrimidin-4-amine
(1S,5R)-3-(2-amino-6-methylpyrimidin-4-yl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[4-(4-ethoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
3-[benzyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
ethyl 7-[methyl(1,3-thiazol-2-ylmethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
2-amino-4-(4-hydroxy-3-methoxyphenyl)-6-(2,4,5-trifluorophenyl)pyridine-3-carbonitrile