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N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)propanamide
5-(1H-imidazol-4-yl)-4-phenyl-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-imidazole
6-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-cyclopropanecarbonyl-2-[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]piperidine
4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-(4-fluorophenyl)piperazin-2-one
N-[2-(methylsulfanyl)ethyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-butyl-8-(2-methyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-{4-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
2-methyl-3-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)quinoxaline
3-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-1-methyl-1H-pyrrole-2-carboxamide
1-cyclopentyl-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-2-one
N-cyclopropyl-N-(1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)furan-2-carboxamide
2-(4-chloro-2-methylphenoxy)-1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}ethan-1-one
{3-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-oxopropyl}urea
N-[2-(2-methoxyphenyl)ethyl]-6-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N-[furan-2-yl(phenyl)methyl]-3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
3-(4-{[4-(3-methylphenyl)phenyl]carbamoyl}piperidine-1-carbonyl)pyridin-1-ium-1-olate
4-{2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]ethyl}benzene-1-sulfonamide
7-(3-methoxypropyl)-2-[2-(methylsulfanyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
5-{4-[(4-cyclopropanecarbonyl-1,4-diazepan-1-yl)methyl]phenoxy}-1-azabicyclo[3.2.1]octane
N-(5-chloro-2-methoxyphenyl)-3-[1-(1H-1,2,4-triazole-5-carbonyl)piperidin-3-yl]propanamide
7-methyl-3-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
methyl 2-{8-[(1-methyl-1H-indol-3-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
N-ethyl-5-[4-(2-phenylethyl)piperazine-1-carbonyl]pyrimidin-2-amine
8-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3,4-dimethylphenyl)methyl]-4-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperazin-2-one
N-butyl-3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-[(2-methylphenyl)methyl]propanamide
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-N-(2,4-dimethoxyphenyl)propanamide
3-(1H-imidazol-2-yl)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidine
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methyl-6-propylpyrimidine
4-(4-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
6-(3-fluoro-4-methoxyphenyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(oxolan-2-ylmethyl)-3-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl}propanamide
methyl 1-[3-(2-aminoethyl)piperidine-1-carbonyl]cyclopropane-1-carboxylate
5-(2,4-dimethoxyphenyl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1,2,4-triazin-3-amine
5-{1-[2-(furan-2-yl)ethyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)-1,3-thiazole
4-(2,4-dioxoimidazolidin-1-yl)-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}benzamide
5-methoxy-2-{[methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenol
4-[(1-ethylpyrrolidin-2-yl)methyl]-6-fluoro-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
3-fluoro-N-{1-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
4-chloro-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[5-(azepane-1-carbonyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]cyclobutanecarboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-[2-chloro-5-(morpholin-4-yl)phenyl]-1-[2-(pyridin-4-yl)ethyl]urea
4-chloro-N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-2-methylbenzamide