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N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-5-methylthiophene-2-carboxamide
6-[(1-methylpiperidin-4-yl)amino]-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
methyl (2S,4R)-4-(4-methylbenzamido)-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidine-2-carboxylate
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1-[(6-chloropyridin-2-yl)methyl]-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
4-hydroxy-N-[(3S)-2-oxoazepan-3-yl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
3-[(1-ethylpyrrolidin-3-yl)methyl]-1-(4-methoxy-2-methylphenyl)urea
3-[(4aR,7aS)-4-{imidazo[1,2-a]pyridin-2-ylmethyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}acetamide
4-(4-fluorophenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-oxobutanamide
N-[(2-chloro-6-fluorophenyl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-benzyl-4-(3,6-dimethylpyrazin-2-yl)-1,4-diazepan-6-ol
N-[2-(2-chlorophenyl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
methyl 3-(2,3-dihydro-1-benzofuran-2-carbonyl)-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(furan-2-ylmethyl)-5-(4-methylpiperidine-1-carbonyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
6-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]pyridine-3-carboxamide
3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-2-(methylsulfanyl)pyridine
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-ethyl-N-(oxolan-2-ylmethyl)acetamide
N,2-dimethyl-N-[(5-methylfuran-2-yl)methyl]oxolane-2-carboxamide
8-(1-benzothiophen-2-ylmethyl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-benzoyl-6-methyl-5-[5-(1H-pyrazol-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
5-(2-{[(5-propyl-1,2-oxazol-3-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxamide
4-(4-{[3-(furan-2-yl)-3-phenylpropyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
3-(2-methylphenyl)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-3-ol
4-[(3-chlorophenyl)methyl]-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
1-[(3,4-dimethylphenyl)methyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
3-(4-fluorophenyl)-6-[3-(1-methoxyethyl)phenyl]pyridazine
{2-[4-(3-fluorophenoxy)piperidin-1-yl]-8-methylquinolin-3-yl}methanol
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-4-(pyridin-4-yl)pyrimidin-2-amine
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-(thiophen-2-ylmethyl)propanamide
1-[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
(1S,6R)-9-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
4-oxo-N-{1-[2-oxo-2-(4-phenyl-1,4-diazepan-1-yl)ethyl]-1H-pyrazol-4-yl}-4-phenylbutanamide
(1S,5R)-3-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-4-(cyclopropylmethyl)-1,4-diazepane-6-carboxylic acid
8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-N-methylbenzamide
1-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
(4aR,7aS)-1-[2-(dimethylamino)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}-2,1,3-benzothiadiazole
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
N-cyclopropyl-2-{[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]amino}pyridine-4-carboxamide
3-({5-[1-(4-methylphenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
2-chloro-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-acetamidobenzamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
methyl 3-{[(3-ethyl-1-methyl-1H-pyrazol-5-yl)formamido]methyl}-5-(furan-2-amido)benzoate
1-(3-oxo-3-{4-[3-oxo-3-(4-phenylpiperazin-1-yl)propyl]piperidin-1-yl}propyl)pyrrolidin-2-one
2-[2-(1H-pyrazol-1-yl)ethyl]-1-(1H-pyrrole-2-carbonyl)piperidine