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N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,3,6-trimethyl-1-benzofuran-2-carboxamide
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(2-phenyl-1,3-thiazol-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(1-methyl-1H-pyrrol-2-yl)-N-[(4-phenylmorpholin-2-yl)methyl]-1H-pyrazole-5-carboxamide
methyl 1-[(3S,5S)-1-[(4-ethoxyphenyl)methyl]-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-{4-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]phenyl}-3-{[1-(hydroxymethyl)cyclopropyl]methyl}-3-methylurea
6-(propan-2-yl)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrimidin-4-amine
(1R,5S)-6-(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)-6-azabicyclo[3.2.1]octane
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-[3-(pyridin-3-yloxy)propyl]propanamide
1-[2-methoxy-4-({[2-(thiophen-2-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N-[(3S,4R)-1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-{4-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]phenyl}acetamide
3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2,5-dimethylpyrazine
2-{[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]methyl}benzonitrile
1-(furan-2-ylmethyl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1,2-oxazol-3-ylmethyl)acetamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
N-(1-{1-[2-(piperidin-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
4-[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl]-1-phenylpiperazin-2-one
(2S,4R)-N-(1-benzothiophen-2-ylmethyl)-N-methyl-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
N,2-dimethyl-N-(quinolin-6-ylmethyl)-1H-imidazole-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
(1S,5R)-3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-ethyl-4-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,2-dihydropyridin-2-one
2-(2-oxopyrrolidin-1-yl)-N-[(3R,4S)-4-(propan-2-yl)-1-(1,3-thiazol-4-ylmethyl)pyrrolidin-3-yl]acetamide
2-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyridine-4-carboxamide
2-[4-(4H-1,2,4-triazol-4-ylmethyl)-1,3-thiazol-2-yl]pyrazine
2-(4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)ethan-1-ol
(3R,4R)-3-methyl-1-[1-(4-methylphenyl)cyclopropanecarbonyl]-4-(oxan-4-yl)piperidin-4-ol
3-acetamido-N-(2-methoxyphenyl)-5-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-4-pentanamidobenzamide
4-(1H-imidazol-2-ylmethyl)-1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-N,N-dimethylaniline
N-(2-fluoro-4-methylphenyl)-2-[(1-phenyl-1H-1,2,3-triazol-5-yl)formamido]acetamide
3-methyl-1-(1-{6-[(piperidin-4-yl)amino]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
N-methyl-2-oxo-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,2-dihydroquinoline-4-carboxamide
4-(1-{1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}benzamide
3-methyl-7-{6-[(propan-2-yl)amino]pyrimidin-4-yl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(2S,4S)-4-{[(2,5-difluorophenyl)methyl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
(2S)-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)piperidine-2-carboxamide
1-(cyclohexylmethyl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-6-oxopiperidine-3-carboxamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-7-acetamido-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazole-5-carboxamide
2-{[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyrimidin-4-yl}-2-ethoxybenzoic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-(3,3,3-trifluoropropyl)-1,4-diazepan-6-ol
1-(azocan-1-yl)-3-[2-methoxy-4-({[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-ethyl-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-methyl-1H-pyrazole-5-carboxamide