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2-(dimethyl-1,2-oxazol-4-yl)-2-[(furan-2-ylmethyl)(methyl)amino]acetic acid
4-benzyl-3-ethyl-1-(3-methoxypyridine-2-carbonyl)-1,4-diazepan-5-one
4-[3-(3-phenylphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]morpholine
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-[1-(2-phenoxyacetyl)piperidin-4-yl]imidazolidine-2,4-dione
3-(3-hydroxypyrrolidine-1-carbonyl)-1-methyl-1,2-dihydroquinolin-2-one
4-cyano-1-methyl-N-[(1R,2S)-2-phenylcyclohexyl]-1H-pyrrole-2-carboxamide
N-(4-fluoro-2-methylphenyl)-3-{1-[2-(1H-imidazol-4-yl)acetyl]piperidin-3-yl}propanamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
N-benzyl-5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}pyrimidin-2-amine
4-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}phenol
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-(dimethyl-1H-1,2,4-triazol-3-yl)urea
2-{3-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
2-hydroxy-4-(methylsulfanyl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]butan-1-one
1-cyclopentyl-4-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-2-one
3-butyl-4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-methylpiperazin-2-one
3-[(2-fluorophenyl)formamido]-N-[2-(1H-imidazol-4-yl)ethyl]propanamide
9-(6-amino-2-methylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
(3S)-4-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
(3S,5R)-1-benzyl-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
ethyl 3-[(3-methoxyphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-3-carboxylate
N-({5-[(2,4,6-trimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-cyclobutanecarbonyl-N-[2-(pyrazin-2-yl)ethyl]piperidine-4-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-(quinolin-6-ylmethyl)piperazin-2-yl}ethan-1-ol
3-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
3-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1-(2-phenylethyl)urea
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-methyl-4-oxo-4H-pyran-2-carboxamide
N-[7-(4-ethylpiperazine-1-carbonyl)-1-(2-phenylethyl)-1H-1,3-benzodiazol-5-yl]-2-methoxyacetamide
N-[2-(diethylamino)ethyl]-2-ethyl-7-(2-methoxybenzamido)-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]acetamide
[2-methoxy-5-(quinolin-3-yl)phenyl]methanol
2-[(2,3-dimethoxyphenyl)methyl]-4-{4-[2-(naphthalen-1-yl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-ethyl-5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}pyrimidin-2-amine
(4aS,7aR)-1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)methanesulfonamide
4-(butane-1-sulfonyl)-9-(cyclopropylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)[(2-phenyl-1,3-thiazol-5-yl)methyl]amine
(1R,5R)-6-benzyl-3-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
6-(benzyloxy)-1-cyclohexyl-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1,4-diazepan-2-one
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-3-(1H-pyrazol-4-yl)benzamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(5-methyl-1,3-oxazole-4-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-[1-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-2-yl]-2-(methoxymethyl)pyrimidine
4-(3-chlorophenyl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-N-{2-phenyl-1-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]ethyl}furan-2-carboxamide
2-(cyclopropylmethyl)-N-(3-ethylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
1-(3-benzoylpiperidin-1-yl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-(2,3-dihydro-1H-inden-5-yl)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
1-(1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-4-yl)piperidin-4-ol
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-1-ene-1-carboxamide