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N-(3-hydroxy-2,2-dimethylpropyl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
1-[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)azetidin-3-yl]-3,5-dimethyl-1H-pyrazole
7-[(1-methyl-1H-1,2,3-benzotriazol-4-yl)sulfonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
9-(3-chloro-4-fluorobenzoyl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-3-(1H-pyrazol-1-yl)benzamide
3-methoxy-N,5-dimethyl-N-(quinolin-5-ylmethyl)thiophene-2-carboxamide
3,5-dimethyl-1-(1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}azetidin-3-yl)-1H-pyrazole
N-[2-(pyridin-3-yloxy)phenyl]-1-(thian-4-yl)pyrrolidine-2-carboxamide
1-[(3-chlorophenyl)methyl]-4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-[(2-methoxyphenyl)methyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-({7-[2-(3,4-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-fluorobenzamide
2-(5-fluoro-2-methylphenyl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
1-(5-propyl-1,3,4-oxadiazol-2-yl)-4-(pyridin-3-yl)piperidin-4-ol
(2R,3R)-3-amino-1'-(2,6-dimethoxybenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridin-2-amine
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-2-yl)propan-1-one
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-ethyl-9-(2-hydroxyacetyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(3S)-N-tert-butyl-2-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-(pyridin-2-ylmethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamide
(4aS,7aR)-1-(morpholine-4-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-chlorophenyl)-4-[1-(3,4-difluorobenzoyl)piperidin-3-yl]piperazine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
ethyl 5-{[(3-benzyl-1,2-oxazol-5-yl)formamido]methyl}furan-2-carboxylate
(1S,5R)-3-(1H-1,2,3-benzotriazole-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[4-(benzyloxy)phenyl]methyl}-4-ethyl-1,4-diazepan-5-one
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-[3-(ethylsulfanyl)phenyl]-2-[4-(2-methoxyethyl)piperazin-1-yl]acetic acid
1-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}azocane
4-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
{[2-(azocan-1-yl)pyridin-3-yl]methyl}[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amine
1-(2-fluorophenyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}cyclopropane-1-carboxamide
(1S,5R)-3-{[5-(dimethyl-1,2-oxazol-5-yl)furan-2-yl]sulfonyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-[3-(dimethylamino)-2,2-dimethylpropyl]acetamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(4-methylphenyl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
3-{1-[2-(2-chlorophenyl)acetyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-({[1-(azepan-1-yl)propan-2-yl]amino}methyl)piperidin-1-yl]-2-methylpropan-1-one
(3aR,6aR)-2-(5-methylthiophene-2-carbonyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[3-(piperidin-4-ylmethyl)benzoyl]-1,4-oxazepan-6-ol
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(1,2-oxazol-3-ylmethyl)benzamide
(3S,7S,8aS)-7-{[(4-tert-butylphenyl)methyl]amino}-3-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(2-methoxyethyl)-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylthiophene-3-carboxamide
2-ethyl-8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[5.5]undecan-3-one
N-[(3,4-dimethoxyphenyl)methyl]-N-methyl-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
2-methyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]propanamide
(3aS,7aR)-5-methyl-2-(quinoxaline-6-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-(azonan-1-yl)-N-[(3S)-2-oxoazepan-3-yl]pyridine-2-carboxamide