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2-[methyl(2-phenylethyl)amino]-N-(thiolan-3-yl)-2,3-dihydro-1H-indene-2-carboxamide
5-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-methoxyphenol
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
3-[(1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}piperidin-4-yl)methyl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-({3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-3-methyl-3-[2-(oxan-2-yl)ethyl]urea
N-[2-(7-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
(3S,4R)-1-({5-chloro-2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-4-(hydroxymethyl)piperidin-3-ol
2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-fluorophenyl)-1H-1,2,4-triazol-3-yl]acetamide
methyl 6-(2-{[(4-methoxyphenyl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butane-1,2-dione
3-[(2-fluorophenyl)formamido]-N-[1-(4-methylpyridin-2-yl)propyl]propanamide
6-chloro-N,N-dimethyl-3-{[4-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]azocane
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2-(2-phenyl-1,3-thiazol-4-yl)-N-(pyridin-2-ylmethyl)acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-[(4-methoxyphenyl)methyl]-3-methyl-1,2-oxazole-5-carboxamide
methyl 5-{3-[(1H-indol-2-ylformamido)methyl]piperidin-1-yl}-5-oxopentanoate
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-1H-pyrrole-3-carboxamide
methyl 3-[2-(4-methoxyphenyl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(1H-imidazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-{3,5-dimethyl-4-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
3-({[(3-chloro-2,6-difluorophenyl)methyl]amino}methyl)piperidin-3-ol
N-ethyl-2-(3-fluorophenoxymethyl)-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
8-(2-benzyl-1,3-thiazole-4-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-hydroxy-N-[(3R,4S)-1-[(4-methoxypyridin-2-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
1-({3-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)azetidin-3-ol
6-cyano-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}pyridine-3-carboxamide
1-(4-{[(cyclopentylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
4-{1-[6-(thiomorpholin-4-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
5-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridine-2-carboxylic acid
2-amino-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-4-methylpyrimidine-5-carboxamide
6-(8-methylquinolin-5-yl)pyridine-2-carboxamide
(1S,5R)-6-benzyl-3-[2-(2-hydroxyphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3,5-difluoro-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyridine-2-carboxamide
1-[(2-methoxyphenyl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
1-[2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenyl]ethan-1-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
N-[4-(3-methoxyphenyl)phenyl]-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine-3-carboxamide
3-{1-[2-(2,5-dioxoimidazolidin-4-yl)acetyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-{4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-1-yl}phenol
N-(cyclopropylmethyl)-N-(2-methoxyethyl)-4-(piperidin-3-yl)benzamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2,4,5-trifluorobenzamide
N-methyl-2-(1H-pyrazol-1-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
4-[1-(2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-3-chloropyridine
1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]azocane
1-(4-{[methyl({[2-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}thiophen-2-yl)ethan-1-one