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3-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propanamide
N-[2-(2-ethoxyphenoxy)ethyl]-2-(ethylsulfanyl)-N-methylpropanamide
2-(ethylamino)-N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
1-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-ol
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N,N-diethyl-1-[1-(1H-indol-2-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-[(1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}pyrrolidin-2-yl)methyl]-1H-pyrazole
methyl 3-(furan-3-carbonyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(4aR,8aS)-6-[(3-chlorophenyl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-(1-methyl-1H-pyrazole-5-carbonyl)-3-(4-phenylbenzoyl)piperidine
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-2-fluoro-N-(pyridin-3-ylmethyl)benzamide
3-{1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
6-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-dimethylpyrimidin-4-amine
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]imidazolidine-2,4-dione
9-[(2-aminopyridin-3-yl)methyl]-2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-(methoxymethyl)piperidine
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)propanamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(6-ethoxy-4-methylquinazolin-2-yl)piperidin-4-amine
8-[3-(3,4-dimethylphenyl)propanoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[1-(2,2-dimethylpropyl)-4-[(2-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-{[7-(adamantane-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
2-(4-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}piperidin-1-yl)pyridine-3-carbonitrile
N,N-diethyl-2-{[4-(furan-3-carbonyl)-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}acetamide
1-[4-(6-methylpyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-3-phenylpropan-1-ol
S-{2-[2-(furan-2-yl)-2-oxoacetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-3-hydroxybutane-1-sulfonamido
5-(2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
2-[9-(morpholine-4-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
7-[(4-fluorophenyl)methyl]-2-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
2-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-indole
2-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]-1H-indole
(1R,7S)-3-(2-acetamidoethyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
8-(7-fluoro-2-methylquinoline-4-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-(aminomethyl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-methylpyrimidin-4-amine
1-(5-methyl-1,2-oxazole-3-carbonyl)-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[2-(methylamino)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-(4-ethylpiperazin-1-yl)-3-{3-[({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}amino)methyl]phenoxy}propan-2-ol
1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
1-cyclohexyl-4-[6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-2-one
5-(1-benzoylpiperidin-4-yl)-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-({[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
{1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
4-methyl-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
(1S)-1-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-(1H-imidazol-4-yl)ethan-1-amine
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]propanamide
1-[(1S,5R)-6-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-benzoyl-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
(3-{[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
3,5-dimethoxy-N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
5-[(2-fluoro-4-methoxyphenyl)methyl]-5-{3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one