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N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)acetamide
1-(pyridin-4-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]methylamine
2-[4-methoxy-3-(prop-2-en-1-yl)phenyl]-1H-1,3-benzodiazole-5-carbonitrile
2,5-dimethyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)furan-3-carboxamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
methyl 1-[2-hydroxy-3-(4-{[(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-[2-(4-chlorophenyl)ethyl]-2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetamide
(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-3-(3-phenylpropyl)piperidin-3-yl)methanol
2,5,7-trimethyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}quinoline-4-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(4-methylpentanoyl)piperidine-2-carboxamide
N-[(2-ethoxyphenyl)methyl]-4-oxo-N-(prop-2-en-1-yl)-3,4-dihydroquinazoline-2-carboxamide
3-[2-(dimethylamino)ethyl]-5-[1-(4-methylbenzoyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
methyl 7-oxo-3-(quinolin-8-ylmethyl)-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N,N-diethyl-4-[(2-fluorophenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
1-(cyclohexylmethyl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2,6-dimethyl-N-{1-oxaspiro[4.4]nonan-3-yl}quinoline-4-carboxamide
N'-(2,3-dimethylphenyl)-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]propanediamide
N-(4-{[1-(2-methylpropyl)-2,4-dioxo-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
1-[2-(3,4-dimethoxyphenyl)acetyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[(2-chlorophenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-{[(3S)-3-(3-methoxyphenyl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
2-(dimethylamino)-2-(4-methylphenyl)-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)acetamide
7-methyl-2-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
5-[(3,4-dimethoxyphenyl)methyl]-5-{3-oxo-3-[3-(2-phenylacetyl)piperidin-1-yl]propyl}pyrrolidin-2-one
(3S)-3-ethyl-4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]morpholine
N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
1-[2-(benzyloxy)benzoyl]-1,4-diazepan-6-ol
2-butyl-8-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-({1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-2-yl}methyl)morpholine
2-(4-cyclobutyl-6-methylpyrimidin-2-yl)-8-methyl-2,8-diazaspiro[4.5]decane
2-(4-chlorophenyl)-N-[4-(dimethylamino)phenyl]morpholine-4-carboxamide
1-[4-({4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}methyl)thiophen-2-yl]ethan-1-one
3,5-dimethoxy-N-{[8-(pyridin-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
N-benzyl-N-methyl-2-(1,2-oxazolidine-2-carbonyl)-2,3-dihydro-1H-inden-2-amine
dimethyl[(4-methyl-5-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
3-[(3-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[(2,4-dimethoxyphenyl)methyl]-3-(2-methoxybenzoyl)piperidine
6-[(2-fluorophenyl)methoxy]-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
3-(6-methoxy-2H-1,3-benzodioxol-5-yl)-[1,2,4]triazolo[4,3-a]pyrazine
{4-[(4-chlorophenyl)methyl]-1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}methanol
2-[4-(3,3,5,5-tetramethylcyclohexyl)piperazin-1-yl]pyridine-3-carboxamide
(3aS,6aR)-5-(1,3-benzoxazol-2-yl)-3-[2-(3-chlorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one