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N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3-thiazole-4-carboxamide
2-[2-({4-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)ethyl]-1,3-thiazole-4-carboxylic acid
N-[(3-fluorophenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-(3-methoxyphenoxy)ethan-1-one
6-oxo-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[2-(1,2,3-thiadiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
2-{1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidin-2-yl}-1H-1,3-benzodiazole
N-[(2R,3R)-1'-[(2-chloro-4-fluorophenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxyacetamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
ethyl 4-[1-(5-hydroxypyridine-2-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
5-[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
2-(4-chloro-1H-pyrazol-1-yl)-1-[(3S)-3-(dimethylamino)azepan-1-yl]ethan-1-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(pyridin-4-ylmethyl)piperidin-4-ol
(5S,9aS,9bS)-5-(2H-1,3-benzodioxol-4-yl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-[(2-hydroxyphenyl)methyl]-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[2-(trifluoromethyl)benzoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
ethyl 1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
methyl 4-[5-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
2,2-difluoro-N-[2-(4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}morpholin-2-yl)ethyl]acetamide
1-methyl-N-{[8-(2-phenylacetyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-indole-2-carboxamide
4-(4-ethoxy-3-methylphenyl)-N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-oxobutanamide
N-[(3-methyloxetan-3-yl)methyl]-4-phenylbutanamide
2-(4-{[2-(2-hydroxyethoxy)phenyl]methyl}-5-methyl-2-oxopiperazin-1-yl)benzonitrile
2-(pyridin-3-yl)-N-[1-(thiophen-3-yl)propan-2-yl]pyrimidine-5-carboxamide
(3R,4S)-4-cyclopropyl-1-[4-(piperidin-1-yl)benzoyl]pyrrolidin-3-amine
2-({[2-(2-ethoxyphenoxy)ethyl](methyl)amino}methyl)-3-methoxyphenol
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
5-(methoxymethyl)-N-[4-(5-methyl-4-{[2-(morpholin-4-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]furan-2-carboxamide
3-methyl-4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
1-(2-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-4-fluorophenyl)-1H-pyrazole
3-(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-2-yl)pyridine
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl({[1-(2-methylpropyl)piperidin-4-yl]methyl}){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-{[3-(cyclopentyloxy)phenyl]methyl}-4-(pyridin-3-yl)piperazine
methyl (2S)-1-{3-[(4-ethylphenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}pyrrolidine-2-carboxylate
(4aR,6R,8aS)-2-(5-chloropyridin-2-yl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-[3-(trifluoromethyl)benzoyl]-6-azaspiro[2.5]octane
5-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)-2-hydroxybenzoic acid
(2S,4S)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-ethyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
N-(1-benzothiophen-5-ylmethyl)-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methoxypyrimidin-4-amine
ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](2-phenylpropyl)amine
1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(piperidin-1-ylmethyl)piperidine
4-(1H-pyrazol-3-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
methyl 1-[(3S,5S)-1-[(2-ethoxyphenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(pyrrolidin-1-yl)pyridazine
1-[(3R,4R)-4-[2-(5-tert-butyl-1H-pyrazol-3-yl)-1H-imidazol-1-yl]oxolan-3-yl]piperidine
1-methyl-5-[3-methyl-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]-1H-pyrrole-3-carbonitrile
9-methoxy-7-(2-methoxyphenyl)-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine