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1-[(2-chlorophenyl)methyl]-5-(2-{[(3-methylphenyl)methyl]amino}ethyl)pyrrolidin-2-one
2-{1-[(1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-amine
N-[2-(4-chlorophenoxy)ethyl]-N-ethyl-4-(1H-pyrazol-3-yl)benzamide
(3aS,6aS)-2-(2-hydroxyethyl)-5-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-({4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}methyl)-N-[1-(naphthalen-1-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-ethyl-6-methyl-5-[5-(4-methyl-1,3-thiazol-5-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
N-(4-methoxy-2-methylphenyl)-3-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-3-yl}propanamide
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazole
4-[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-6-(pyrrolidin-1-yl)pyrimidine
4-(propan-2-yl)-6-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrimidin-2-amine
2-{1-cyclohexyl-4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-[(4-{[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}-6-methylpyrimidin-2-yl)amino]phenol
N-butyl-N-[(3-methylthiophen-2-yl)methyl]-1-(oxan-4-yl)piperidine-4-carboxamide
methyl 3-(4-{1-[N-methyl-2-(1H-pyrazol-1-yl)acetamido]-2-phenylethyl}piperidine-1-carbonyl)benzoate
3-{4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
2-(1-{5-[(dimethylamino)methyl]-1,3,4-oxadiazole-2-carbonyl}piperidin-3-yl)propan-2-ol
1-(2-methoxyethyl)-8-[(4-methoxyphenyl)methyl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxybenzoyl)piperazine
2-cyclopentyl-8-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(1H-imidazol-2-ylmethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
3-[({1-[2-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)methyl]pyridine
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(3-phenylphenyl)methyl]pyrrolidin-3-yl]methanol
2,5-dichloro-N-{2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxoethyl}benzamide
2-(3,5-difluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3aS,6aS)-2-[(4-phenoxyphenyl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(2,2-dimethylpent-4-en-1-yl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-({3-[3-(2-methoxyphenyl)phenyl]-1H-pyrazol-1-yl}methyl)-5-methyl-1,2,4-oxadiazole
1-methyl-2-oxo-8-(phenylcarbamoyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[3-(3-ethylphenoxy)azetidin-1-yl]-2-hydroxy-2-(4-methoxyphenyl)ethan-1-one
8-(3-aminopropanoyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1H-imidazol-4-ylmethyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
methyl 8-[(2,5-dimethoxyphenyl)methyl]-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-cyclohexyl-N-methyl-3-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
methyl N-({[(3R,5S)-5-(ethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]carbamoyl}methyl)carbamate
N-methyl-5-{[3-(1-methylpiperidin-3-yl)propanamido]methyl}-1,2,4-oxadiazole-3-carboxamide
ethyl 5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(dimethylamino)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
({6-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyrazin-2-yl}methyl)dimethylamine
1-(cyclopropanesulfonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(1S,5R)-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(benzyloxy)-8-(3-fluoro-4-methoxybenzoyl)-1,8-diazaspiro[4.5]decan-2-one
N-(adamantan-2-ylmethyl)-5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]propanamide
1-(2-methoxypyridine-4-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
(3S,4S)-4-cyclopropyl-1-[4-(1H-pyrazol-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
2-{2-[(3-methylpyridin-2-yl)amino]ethyl}-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(4-ethoxyphenyl)propyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
(3R,5R)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
2-{[(2-methylphenyl)methyl]sulfanyl}-N-(1H-1,2,4-triazol-5-ylmethyl)acetamide