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4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]pyrimidin-2-amine
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(piperidin-1-ylmethyl)piperidine
4-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(2-fluorophenyl)pyrimidine
4-{1-[3-(dimethylcarbamoyl)propanoyl]piperidin-3-yl}benzoic acid
2-[4-(6-methoxyquinolin-3-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
5-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
4-{1-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-2-methylpropan-2-yl}morpholine
8-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-(furan-2-ylmethoxy)phenyl]-3-[2-(piperidin-1-yl)ethyl]urea
2-[1-cyclohexyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
ethyl 1-{6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carbonyl}piperidine-3-carboxylate
4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N-methylpyridin-2-amine
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
8-chloro-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)quinoline-2-carboxamide
4-(3,3-dimethylpyrrolidine-1-carbonyl)-6-fluoro-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
N-{3-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]phenyl}acetamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-{[3-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]methanol
N-(1-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
1-(cyclopropylmethyl)-N-(3,4-difluorophenyl)piperidin-3-amine
3-{2-[1-butyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
2-(adamantan-1-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
5-acetyl-N-cyclopropyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]thiophene-3-carboxamide
N-[(5-methylthiophen-2-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(2,5-difluorobenzoyl)piperidin-1-yl]ethan-1-one
N-[(3S,4R)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-(dimethylamino)-3-(4-methoxy-2-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}phenoxy)propan-2-ol
2-(3-hydroxypropyl)-9-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-fluoro-2-(3-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
1-[(4-chlorophenyl)methyl]-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(2-chlorophenyl)-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}acetic acid
3-amino-1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}pyrrolidine-3-carboxylic acid
4-methoxy-N-(2-methoxyethyl)-2-[(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)oxy]benzamide
N-[(3S)-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
4-(2-fluorophenoxy)-1-(furan-3-carbonyl)piperidine-4-carboxylic acid
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2,4-dimethylpyrimidine-5-carboxamide
3-[2-({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
4-[(4-methyl-5-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
1-(3-carbamoylpropanoyl)-N-[3-(4-fluorophenyl)phenyl]pyrrolidine-2-carboxamide
1-[2-(dimethylamino)ethyl]-6-oxo-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
N-ethyl-3-(2-phenylethyl)piperidine-1-carboxamide
methyl 3-[(4-benzoyl-7-oxo-1,4-diazepan-1-yl)methyl]benzoate
4-chloro-1-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-1,3-benzothiazole-6-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-3-ol
1-methyl-3-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)-3-(4-phenylphenyl)pyrrolidine-2,5-dione
3,5-dichloro-4-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
1-cyclohexyl-N3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide