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2-(3-hydroxypropyl)-9-(3,3,3-trifluoro-2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
[(1-benzylpiperidin-4-yl)methyl](methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-[1-(cyclohex-1-en-1-yl)ethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
4-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
2-(methylamino)-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-1,3-thiazole-4-carboxamide
2-methyl-1-[1-(3-methylthiophene-2-carbonyl)azetidin-3-yl]piperidine
5-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-2-(propylsulfanyl)pyrimidine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(propan-2-yloxy)benzamide
1-(4-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}piperidin-1-yl)ethan-1-one
3-[(2-methyl-1H-imidazol-1-yl)methyl]-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidine
3-ethyl-6-(7-fluoro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-3H-imidazo[4,5-b]pyridin-2-amine
(2S,4R)-4-[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
9-{[4-(2-aminoethyl)phenyl]methyl}-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6-phenyl-3-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-dihydropyridin-2-one
3-({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
3-[1-(ethanesulfonyl)piperidin-4-yl]-N-(2-methoxyethyl)propanamide
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]urea
2-(3-chloro-4-ethoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-4-(1H-pyrazol-1-yl)benzamide
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(5-fluoro-2-methylphenyl)methyl]acetamide
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
2-(2-fluoro-5-methoxyphenyl)-5-methyl-4-[(4-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(oxan-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-methylfuran-2-carboxamide
5-methyl-4-{[2-(morpholin-4-yl)ethyl]amino}-N-[3-(propan-2-yloxy)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-(5-methanesulfonamido-2-methylphenyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
{1-[(5-ethylfuran-2-yl)methyl]-4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
(1R,3S)-3-ethoxy-7-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-7-azaspiro[3.5]nonan-1-ol
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-N-(2-phenylethyl)piperidin-3-amine
5-{3-[3-(3-methylbutanoyl)piperidin-1-yl]-3-oxopropyl}-5-(naphthalen-1-ylmethyl)pyrrolidin-2-one
3-[(3R,4S)-1-[2-(2-methoxyphenyl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[3-(thiophene-2-carbonyl)piperidin-1-yl]butan-1-one
4-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}-3-methyl-1-(prop-2-en-1-yl)-1H-pyrazole
{2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
3-(2-fluorophenyl)-5-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
6-[methyl(propan-2-yl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-[methyl(pyridin-2-ylmethyl)amino]-1-[3-(pyridin-4-yl)azetidin-1-yl]ethan-1-one
3-[3-(1H-imidazol-1-yl)propyl]-1-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
methyl 2-chloro-5-{[4-(4-methoxybutyl)piperazine-1-carbonyl]amino}benzoate
3-{[2-(2-aminoethyl)quinazolin-4-yl]amino}-N-(2-ethylphenyl)propanamide
1-benzyl-4-{2-[2-(furan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}pyrrolidin-2-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-5-methyl-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-butyl-4-{[(3-fluorophenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-(3-methoxypropyl)-1-{[5-(3-methyl-1,2-oxazol-5-yl)furan-2-yl]sulfonyl}piperidine
1-[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-3-yloxy)ethan-1-one