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(2S,4S)-4-(4-{[2-(4-fluorophenyl)acetamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
5-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
2-{4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]morpholin-3-yl}acetic acid
N-(1-cycloheptylpiperidin-3-yl)-3-(2-fluorophenyl)-1H-pyrazole-4-carboxamide
5-(2,6-dimethylphenoxymethyl)-N-(prop-2-en-1-yl)-1,2-oxazole-3-carboxamide
2-chloro-N-[5-(2-ethylpiperidine-1-carbonyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-6-fluorobenzamide
2-[6-(dimethylamino)pyridine-3-carbonyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1-methylcyclohexane-1-carboxamide
N-(2-phenylethyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-amino-4-[4-(3-hydroxyprop-1-yn-1-yl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-4-(1H-pyrrol-1-yl)benzamide
4-ethyl-3-{[1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{1-ethyl-7-[4-(2-methoxyethyl)piperazine-1-carbonyl]-2-(pyridin-3-yl)-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
4-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]butanamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carboxylic acid
4-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}-5-methoxypyridin-4-ol
1-{3-[(3-{[3-(dimethylamino)propyl](methyl)amino}piperidin-1-yl)methyl]phenyl}ethan-1-one
4-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
methyl 2-[8-(naphthalen-1-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
methyl (2S,4S)-1-[(4-ethoxyphenyl)methyl]-4-(naphthalene-1-amido)pyrrolidine-2-carboxylate
1-[(4-methoxyphenyl)methyl]-4-[2-(pyridin-3-yl)acetyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-4-methoxy-N-(pyridin-3-ylmethyl)benzamide
6-[(3-methoxyphenyl)methoxy]-4-(oxolane-3-carbonyl)-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
3-(4-methoxyphenyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]pyrrolidin-3-yl]acetamide
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
methyl 3-(3-methylthiophene-2-carbonyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(2,3-difluorobenzoyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)naphthalene-1-carboxamide
ethyl 1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)piperidin-3-ol
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
(2-methoxyethyl)({1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-2-phenylethyl})(pyridin-3-ylmethyl)amine
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2,6-dimethylpyrimidine-4-carboxamide
[3-(3-methylbut-2-en-1-yl)-1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-3-yl]methanol
6-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-ylmethyl}quinoline
3-(1-ethoxypropyl)-4-[(3-fluorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aS)-2-(dimethylcarbamoyl)-5-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[3-(dimethylamino)propyl]-9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(benzenesulfonyl)pyrrolidin-3-yl]methanol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(6-methylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[5-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
5-{1-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-methylpropyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
1-ethyl-N-methyl-3-(pyrrolidine-1-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-ethyl-2-(morpholin-4-yl)-N-[2-(pyridin-2-yl)ethyl]pyrimidin-4-amine
N-methyl-N-[1-(pyridin-2-yl)ethyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(2-fluorophenyl)propan-1-one
2-(dimethyl-1,2-oxazol-4-yl)-1-(3-{5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)ethan-1-one