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8-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(2,2-dimethyloxan-4-yl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
methyl 2-[N-methyl-3-(2-methylphenyl)-3-phenylpropanamido]acetate
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
6-(3-chlorophenyl)-N-[(2-methoxyphenyl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(4-methoxyphenoxymethyl)-6-(1-methylpiperidin-4-yl)-3,4-dihydropyrimidin-4-one
4-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1-(1H-indazol-5-yl)piperazin-2-one
(1S,5R)-6-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
1-cyclopropyl-6-oxo-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]piperidine-3-carboxamide
1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-3-(2-methoxybenzoyl)piperidine
1-[(5-ethylfuran-2-yl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
methyl 1-[(3R,5S)-5-[(diphenylmethyl)carbamoyl]-1-(quinolin-6-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-acetamido-N-(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)pyrrolidine-1-carboxamide
8-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}quinoline-2-carboxamide
7-(propan-2-yl)-2-(pyridine-3-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{2-[2-(3-methoxyphenyl)-1H-imidazol-1-yl]ethyl}pyridine-4-carboxamide
3-{2-[2-(3-fluorophenyl)azepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-(2-chlorophenyl)-4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
3-(2-chlorophenyl)-1-[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-phenylethyl)piperidin-1-yl]propan-1-one
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(oxolan-3-ylmethyl)piperazine
N-[(3S,5S)-5-{[2-(1H-imidazol-4-yl)ethyl]carbamoyl}-1-methylpyrrolidin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5,5-diphenylpiperidin-2-one
2-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}thieno[3,2-d]pyrimidin-4-amine
1-[4-(2-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}-2-oxoethyl)phenyl]imidazolidin-2-one
1-[2-(1-benzothiophen-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine-3-carboxamide
3-(1-methyl-1H-pyrazol-5-yl)-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
(3S,4S)-1-(1-methyl-1H-pyrazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-6-methylpyridine-2-carboxamide
1-ethyl-N-[(1-hydroxycyclohexyl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-1-(propan-2-yl)piperidine-4-carboxamide
2-{4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-1-yl}-1,3-benzothiazole
methyl 3-[(3S,4R)-1-[(2-hydroxy-4-methoxyphenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
N-[(2R,3R)-2-methoxy-1'-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
3-fluoro-N-(1-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
methyl 1-(2-methoxyethoxy)-2-oxo-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
N-({8-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-fluorobenzamide
3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
N-phenyl-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-amine
2-(1,4-diazepane-1-carbonyl)-6-(2,5-dimethylfuran-3-yl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-{1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}methanesulfonamide
7-methoxy-3-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
ethyl 1-ethyl-5-(1-ethyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-methyl-4-({8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-1H-pyrrole-2-carbonitrile
8-methoxy-2-(4-methoxy-3-methylphenyl)-5-[(4-methyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
benzyl({[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl})methylamine
1-(cyclopropylmethyl)-N-methyl-5-(naphthalen-1-ylmethyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(4-acetyl-1,4-diazepan-1-yl)-2-(6-methoxynaphthalen-2-yl)acetic acid