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1-(ethanesulfonyl)-4-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}piperazine
3-(4-methylphenyl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-3-phenylpropanamide
2-methoxy-4-[4-(3-methylpyridin-2-yl)piperazin-1-yl]pyridine-3-carbonitrile
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
6-{3-oxo-3-[4-(piperidine-1-carbonyl)piperidin-1-yl]propyl}-2,3-dihydropyridazin-3-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
6-(3-chlorophenyl)-7-(cyclopropylmethyl)-N-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(1-methyl-1H-pyrazol-5-yl)-1-[4-(pyridin-4-yl)piperazin-1-yl]propan-1-one
2-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
N-(thiophen-3-ylmethyl)-9H-purin-6-amine
N-(2-methyl-1-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
4-phenyl-N-({1-[2-(pyridin-3-yl)acetyl]piperidin-3-yl}methyl)benzamide
8-(4-amino-3-hydroxybutanoyl)-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(4-methoxyphenyl)-4-[1-(2-phenylethyl)piperidin-3-yl]piperazine
7-(3-chlorophenyl)-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,7S)-5-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-methyl-4-[4-({4-[(methylsulfanyl)methyl]piperidin-1-yl}methyl)phenyl]butan-2-ol
N-[2-(morpholin-4-yl)ethyl]-5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2-hydroxyphenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-methyl-N-(oxolan-3-yl)-1,3-oxazole-4-carboxamide
[(4-{2-[1-(3-chlorobenzoyl)piperidin-2-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
(4aR,7aS)-1-ethyl-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{3-oxo-3-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propyl}azepan-2-one
1-(2-{4-[benzyl(methyl)amino]piperidin-1-yl}-2-oxoethyl)azepan-2-one
4-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{[1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,3-benzothiazole
2-(3,5-dimethyl-1H-pyrazol-4-yl)-5,6-dimethylpyridine-3-carboxamide
3-[1-(3-propyl-1H-pyrazole-5-carbonyl)azetidin-3-yl]pyridine
4-cyclohexyl-N-(3-methanesulfonamidophenyl)piperazine-1-carboxamide
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
4-fluoro-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
(1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
4-(6-fluoro-2-methylquinolin-4-yl)benzamide
(2S,4R)-N-(1-benzothiophen-2-ylmethyl)-N-methyl-1-[(3-methylphenyl)methyl]-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
11-[(9H-fluoren-9-yl)amino]-4-[2-(pyridin-2-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 6-(4-fluorobenzoyl)-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-chloro-4-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-dimethyl-1H-pyrazole
1-[1-ethyl-5-(2,4,5-trifluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methylbenzamide
5-(hydroxymethyl)-2-methyl-4-({methyl[1-(2-phenylethyl)piperidin-3-yl]amino}methyl)pyridin-3-ol
5-ethyl-3-[(2-{2-phenylimidazo[1,2-a]pyridin-3-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)(quinolin-4-ylmethyl)amine
N-(2-methyl-1-{7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)methanesulfonamide
4-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-N,N-dimethylpiperazine-1-carboxamide
1-[5-tert-butyl-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
4-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyrimidin-2-yl}morpholine
2-(1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)ethan-1-ol
1-{2-[2-(butan-2-yl)phenoxy]acetyl}piperidine-4-carboxylic acid