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1-(3-chloro-4-hydroxybenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-chloro-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylthiophene-2-carboxamide
2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(trifluoromethyl)pyridine
1-{7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-3-propoxypiperidine
N-{4-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}carbamoyl)methyl]phenyl}butanamide
methyl (2S)-2-{[5-(3-methoxyphenoxymethyl)-1,2-oxazol-3-yl]formamido}-3-methylbutanoate
1-(4-methoxybenzoyl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazine
7-[(4-fluorophenyl)methyl]-2-(1-phenyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
N3-butyl-N5-[(3-fluoro-4-methylphenyl)methyl]-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
6-[1-(3-methylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
(2E)-N-({3-methyl-7-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
8-(5-chloro-3-fluoropyridin-2-yl)-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-[1-(2,3-dihydro-1H-inden-4-yl)-5-[(2,4-dioxoimidazolidin-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
4-(3-methoxypropyl)-1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
methyl 1-({4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-2-carboxylate
N-benzyl-N-(cyclobutylmethyl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-imidazole-2-carboxamide
5-[4-(4-methoxypyrimidin-2-yl)piperazine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(pyridin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[2-(morpholin-4-yl)pyridin-3-yl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-hydroxy-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrazine-2-carboxamide
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine
3-(5-{[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decane
methyl 3-(2-methoxybenzamido)-5-{[(4-methyl-1,3-oxazol-5-yl)formamido]methyl}benzoate
1-[3-(3-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}phenoxy)propyl]-1H-imidazole
5-benzamido-1-cyclopentyl-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-1,3-benzodiazole-7-carboxamide
1-(4-cyanophenyl)-3-{1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}urea
2-(3-methoxyphenyl)-1-{4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
(2S,4S)-4-amino-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methylpyrrolidine-2-carboxamide
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
3-({4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
N-[1-(4-methoxyphenyl)ethyl]-N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[2-(4-fluorophenyl)ethyl]benzamide
[4-(naphthalen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl](pyridin-3-yl)methanol
N-[1-(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]pyridine-2-carboxamide
methyl (2S,4R)-4-(dimethylamino)-1-[2-(pyridin-4-yl)ethanesulfonyl]pyrrolidine-2-carboxylate
(3S,4R)-1-[3-(2-oxopyrrolidin-1-yl)benzoyl]-4-phenylpyrrolidine-3-carboxylic acid
1'-(4-methyl-1H-imidazole-2-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]
5-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide
2-(2,3-dihydro-1-benzofuran-7-yl)-5-fluoro-4-methoxypyrimidine
(2R)-N-[2-(dimethylamino)ethyl]-2-methoxy-N-[(3-methylthiophen-2-yl)methyl]-2-phenylacetamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
4-{4-[2-(methylamino)pyridine-4-carbonyl]piperazin-1-yl}butan-1-ol
5-ethyl-2,3-dimethyl-N-[2-(1,3-thiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamide
(3aS,6aS)-2-methyl-5-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-chloro-3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}urea