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methyl 3-(furan-2-amido)-1-(2-methoxyethyl)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methyl-N-(oxan-4-ylmethyl)acetamide
(2,1,3-benzoxadiazol-5-ylmethyl)({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
2-methyl-2-[2-(4-methyl-1,4-diazepan-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]propanoic acid
N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)propanamide
3-(oxolan-3-yl)-5-(3-phenoxyphenyl)-1,2,4-oxadiazole
3-(5-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}thiophen-2-yl)-1H-pyrazole
3-(1H-imidazol-1-ylmethyl)-1-[(5-methylthiophen-2-yl)methyl]piperidine
methyl 1-(2-butyl-1,3-benzoxazole-5-carbonyl)piperidine-2-carboxylate
2-(2,4-dimethylphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
2-[3-(cyclopropylmethyl)-5-[(4,5-dimethyl-1H-imidazol-1-yl)methyl]-1H-1,2,4-triazol-1-yl]benzoic acid
N-(2-hydroxyethyl)-1-methyl-N-[(2-methylphenyl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
8-chloro-2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]quinoline
{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amine
N-{[5-(naphthalen-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-methyl-5-({methyl[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)pyrimidin-2-amine
1-methyl-3-({3-oxo-2-azaspiro[4.4]nonan-2-yl}methyl)-1,2-dihydroquinolin-2-one
(2R,3R)-3-({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]pyridine
ethyl 1-[2-(4-ethylpiperazin-1-yl)acetyl]-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
4-methyl-2-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
1-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(1S,6R)-9-(2,3-dimethylquinoxaline-6-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
3-chloro-N-(2-methoxyethyl)-4-({1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}oxy)benzamide
1-[2-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)pyrimidin-4-yl]pyrrolidin-3-ol
1-[(6-methoxypyridin-3-yl)methyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
(4aR,7aS)-4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
benzyl 1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxylate
5-(1-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
7-cyclohexyl-2-(6-methoxypyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 2-[4-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}amino)phenyl]acetate
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-ethyl-2-methylpyrimidin-4-amine
14-(4-butoxyphenyl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
methyl 1-{[4-(2-acetylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-{2,7-diazaspiro[4.5]decan-7-yl}-2-oxoacetamide
(4aS,7aR)-1-[4-(hydroxymethyl)benzoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cycloheptyl-3-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}propanamide
2-methyl-2-[(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]propanamide
[3-(3-phenylpropyl)-1-(quinolin-5-ylmethyl)piperidin-3-yl]methanol
N4-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-2,4-dimethoxybenzamide
2-ethyl-4-methyl-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidine
N-[1-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-methylbutanamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
5-chloro-N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxamide
N-[(3,5-dimethoxyphenyl)methyl]-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide