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N3-ethyl-N1-[2-(2-methoxyethoxy)phenyl]pyrrolidine-1,3-dicarboxamide
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}thiomorpholine
3-methyl-7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-[3-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]piperidine
N-[2-(ethanesulfonyl)ethyl]-3-ethyl-5-hydroxyadamantane-1-carboxamide
4-(benzyloxy)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]butan-1-one
1-[1-(5-ethylthiophene-3-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
3-(2-ethyl-1H-imidazol-1-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylpropanamide
4-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidine
1-({5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)butan-2-ol
1-{1-[2-(1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1-(propan-2-yl)-1H-imidazole
N-(2-{7-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(hydroxymethyl)-N-methylbenzamide
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methoxymethyl)piperidine
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-[1-(pyridin-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[(3R,4S)-1-(4-aminopyrimidin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-4-methylpiperidine-4-carboxamide
N-[(4-hydroxyazepan-4-yl)methyl]-5-methyl-1-benzofuran-2-carboxamide
5-(2,4-difluorophenoxymethyl)-3-(2-methoxyethyl)-1,2,4-oxadiazole
N-[(3R,4S)-1-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]-4-propylpyrrolidin-3-yl]-2-methoxyacetamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)imidazo[1,2-a]pyrimidine-2-carboxamide
(1R,5S,6S)-6-[(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-3-azabicyclo[3.1.0]hexane
(3S,9aR)-3-benzyl-8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{4-[(3,7-dimethyl-1H-indol-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
ethyl(1H-imidazol-2-ylmethyl)({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amine
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,2,3,4-tetrahydroquinazoline-2,4-dione
1-(4-{[cyclohexyl(2-hydroxyethyl)amino]methyl}thiophen-2-yl)ethan-1-one
4-(2-chloropyridine-4-carbonyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-ethyl-2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(oxolan-2-ylmethyl)benzamide
(2S,4S)-N-ethyl-4-[5-(hydroxymethyl)furan-2-amido]-1-(1,3-thiazol-2-ylmethyl)pyrrolidine-2-carboxamide
2-{5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
methyl 2-{1-benzyl-8-[(1-methyl-1H-indol-3-yl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazole
N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyrrolidin-1-yl)benzamide
1-(morpholin-4-yl)-3-(3-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}phenoxy)propan-2-ol
3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
8-(1H-indazole-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-5-(phenoxymethyl)-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-3-carboxamide
1-(3-{4-[3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)phenoxy]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-4-phenylbutan-1-one
3-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
(5S,9aS,9bS)-2-methyl-5-(5-methylfuran-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
{3-[(2-fluorophenyl)methyl]-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl}methanol
N-{3-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-4-methylbenzamide
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl){[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine