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8-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-4-[(dimethylamino)methyl]benzamide
methyl[(4-phenoxyphenyl)methyl]{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
1-{furo[3,2-c]pyridin-4-yl}-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylic acid
1-[(1-benzyl-1H-imidazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
cyclopentyl 4-({[(5-carbamoyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}amino)benzoate
7-[2-(prop-2-en-1-ylsulfanyl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenol
2-(adamantan-1-yl)-4-hydroxy-N-(oxan-3-yl)pyrimidine-5-carboxamide
methyl 5-{[2-(5-cyano-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)acetamido]methyl}furan-2-carboxylate
2-(dimethylamino)-N-methyl-2-(2-methylphenyl)-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[cyclopentyl(methyl)amino]ethan-1-one
3-(2-methylphenyl)-3-[2-oxo-2-(3-propanoylpiperidin-1-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
2-[(3,5-difluorophenyl)methyl]-8-(5-fluoropentyl)-2,8-diazaspiro[4.5]decan-3-one
1-(3-methoxyphenyl)-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperazin-2-one
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
3-(diethylamino)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}propanamide
2-amino-N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-4-methyl-1,3-benzothiazole-6-carboxamide
6-propyl-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(2H-1,3-benzodioxol-5-yl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}acetamide
N-{[3-(2-methoxyethoxy)phenyl]methyl}oxane-2-carboxamide
3-fluoro-N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)benzamide
2-[(4aR,7aS)-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(4-phenylpiperidin-1-yl)ethyl]propanamide
3-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
N-(3-aminopropyl)-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
2-[(4aR,7aS)-6,6-dioxo-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
(3S,4S)-1-(1-methyl-1H-pyrazole-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
4-{2-methyl-6-[1-(oxane-4-carbonyl)piperidin-4-yl]pyrimidin-4-yl}morpholine
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-cyclopropanecarbonyl-5-[(furan-2-ylmethyl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
methyl 4-[2-(4,5-dimethylfuran-2-yl)-1H-imidazol-1-yl]butanoate
2-phenyl-1-(4-{5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidin-4-yl}piperidin-1-yl)ethan-1-one
(3R,4R)-3-cyclobutyl-N-[(3-fluorophenyl)methyl]-3-hydroxy-4-methylpyrrolidine-1-carboxamide
N-{1-[4-(dimethylamino)phenyl]-3-hydroxypropan-2-yl}-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-8-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
N-[(2-{4-[3-(4-methoxyphenyl)propanamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2-phenylpropanamide
3-(1-{imidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)-1-(morpholin-4-yl)propan-1-one
2-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
N-{6-methoxy-2-oxo-4-[1-(propan-2-yl)piperidin-4-yl]-1,2,3,4-tetrahydroquinolin-7-yl}acetamide
N-methyl-N-(2-phenylethyl)-5-{[(pyridin-2-ylmethyl)amino]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[3-(2-oxopyrrolidin-1-yl)propanoyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N-(furan-2-ylmethyl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(but-2-yn-1-yl)-5-(3-phenylpropyl)-5-[1-(pyridin-3-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenylacetamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[2-(methylamino)acetyl]piperidin-4-yl}oxy)benzamide
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-4-carboxylic acid