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3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)propanamide
(3R,4R)-1-[2-(3-methylphenyl)benzoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
(3E)-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}hex-3-en-1-one
(2E)-N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
1-(2-methyl-4-{[2-(3-methylpyridin-2-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
N,N-dimethyl-7-(4-methyl-1H-imidazole-2-carbonyl)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-methyl-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(quinolin-5-ylmethyl)propanamide
1-(1H-indazol-5-yl)-4-[2-(oxan-2-ylmethoxy)acetyl]piperazin-2-one
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-{[2-(trifluoromethyl)phenyl]methyl}cyclopentane-1,3-dicarboxamide
3-(3-hydroxy-3-methylbutyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
3-chloro-2-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
(1S,4R)-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carboxamide
N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
5-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
1-[1'-(4-methoxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-(1-{1-[2-(quinazolin-4-yloxy)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}oxan-4-amine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
5-{1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]piperidin-4-yl}-3-(furan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
4-(3-methoxypropyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 2-chloro-4-({[(1-hydroxycyclohexyl)methyl]carbamoyl}amino)benzoate
1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-amino-4-(4,5-dimethylfuran-2-yl)-6-(pyridine-3-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(4aR,7aS)-1-(2-methoxyethyl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
benzyl[3-(methylsulfanyl)propyl](oxolan-2-ylmethyl)amine
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
(2S)-2-(dimethylamino)-1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-3-phenylpropan-1-one
4-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-2-methylphenol
2-chloro-N-[2-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
2-{[3-(hydroxymethyl)morpholin-4-yl]methyl}-3,5-dimethoxybenzoic acid
N-[2-(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)ethyl]acetamide
N-[2-(4-methylmorpholin-2-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
1-methyl-N-{2-[3-(trifluoromethyl)phenyl]ethyl}azepane-2-carboxamide
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-cyclopropylpyridine-4-carboxamide
N-methyl-N-[2-(2-methylphenyl)-1-[1-(4-phenylbutanoyl)piperidin-4-yl]ethyl]-2-(1H-pyrazol-1-yl)acetamide
2-ethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-(2-chlorophenyl)-7-(2,2-dimethylpropyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(morpholin-4-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(1H-indol-3-yl)ethan-1-one
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-3-cyclopropyl-1H-pyrazole-5-carboxamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methylpyrido[2,3-d]pyrimidin-4-amine
N-{[3-methyl-7-(2,2,3,3-tetramethylcyclopropanecarbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(piperidin-1-yl)acetamide
1-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
3-({[1-(2-methyl-3-phenylcycloprop-2-ene-1-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
[(dimethyl-1,3-thiazol-5-yl)methyl][(1-ethyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
[3-(prop-2-en-1-yl)-1-(pyridine-3-sulfonyl)piperidin-3-yl]methanol