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2-cyclobutyl-1-methyl-7-(oxolane-2-amido)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,3-benzodiazole-5-carboxamide
6-(benzyloxy)-1-cyclohexyl-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
3-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-N,N-dimethylpyrazin-2-amine
2-{4-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}-1,3-benzothiazole
N-(2-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
5-{4-[(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}pyridine-2-carbonitrile
7-(2,3-dimethoxyphenyl)-9-methoxy-4-[(3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(4-benzylpiperazin-1-yl)methyl]-N-cyclohexyl-N-methyl-1,3-oxazole-4-carboxamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-(1,3-dimethyl-1H-pyrazol-5-yl)-3-(2-phenylethyl)-4H-1,2,4-triazole
6-{[methyl(thiophen-3-ylmethyl)amino]methyl}-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide
4-{[2-(acetamidomethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}benzoic acid
N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
(4aR,8aS)-1-(2,2-diphenylethyl)-6-[(4-methoxy-2,5-dimethylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
4-{4-[(2-chloro-6-fluorophenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-(2-{1-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-imidazol-2-yl}phenoxy)ethan-1-ol
7-chloro-4-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-cyclopropyl-9-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-methyl-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
3-{[(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)amino]methyl}piperidin-3-ol
4-[(6-chloro-4-oxo-4H-chromen-3-yl)methyl]-6-methyl-1-(2-methylphenyl)piperazin-2-one
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propan-1-one
methyl 4-[({1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}amino)methyl]benzoate
1-(1'-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(4-fluorophenyl)piperidine
1-{[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
(2S)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-2-phenylethan-1-ol
N-[4-(2-fluorophenoxy)phenyl]-1-(5-methylpyrazine-2-carbonyl)piperidine-2-carboxamide
methyl 1-[5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-yl]piperidine-4-carboxylate
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}ethan-1-one
N-({1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidin-3-yl}methyl)-1H-1,2,4-triazole-5-carboxamide
5-(3-{[(1,4-dithiepan-6-yl)amino]methyl}pyrrolidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
5-{[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-3,4-dihydropyrimidin-4-one
N-[1-(3,4-dimethoxyphenyl)propyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3-methylthiophen-2-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-cyclopropyl-3-[1-(cyclopropylmethyl)piperidin-4-yl]propanamide
2-phenyl-1-(1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)ethan-1-one
3-(but-2-yn-1-yl)-5-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
5-(1-cyclohexyl-4-hydroxypiperidin-4-yl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1-benzofuran-2-carboxamide
2-cyclopentyl-1-[4-(3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]ethan-1-one
1-{3-[4-(benzyloxy)piperidin-1-yl]-3-oxopropyl}azepan-2-one
1-methyl-5-(4-methylpiperidin-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
1-{2-[(2-ethoxyphenyl)carbamoyl]ethyl}-N-methylpyrrolidine-3-carboxamide
(3R,4R)-1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
2-[cyclopropyl(1H-indol-5-ylmethyl)amino]-N-(2-acetamidophenyl)acetamide
N-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidin-4-yl]pyrimidin-2-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(4-hydroxyphenyl)ethan-1-one