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1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-hydroxyethan-1-one
4-(4-methoxy-3-methylbenzoyl)-1-(2-methylphenyl)piperazin-2-one
1-(furan-2-ylmethyl)-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}piperidine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
[3-(1H-imidazol-1-yl)propyl]({[5-(oxan-2-yl)furan-2-yl]methyl})(pyridin-3-ylmethyl)amine
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidine-3-carbonitrile
N-[(4-chlorophenyl)methyl]-1-{2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-[3-(propan-2-yloxy)benzoyl]piperidine
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-cyclopropanecarbonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
(2R,6S)-2,6-dimethyl-4-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}morpholine
1-(4-fluorophenyl)-4-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butane-1,4-dione
(1S,5R)-3-[3-(3-chlorophenyl)propanoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-(furan-2-yl)-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
1-(5-propylpyrimidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-[(4-methoxyphenyl)methyl]-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,2-oxazole-5-carboxamide
1-[3-(1H-imidazol-2-yl)benzoyl]-N,N-dimethylazepan-4-amine
6-[1-(7-chloroquinolin-4-yl)piperidin-4-yl]-2-methylpyrimidin-4-ol
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-(methoxymethyl)-N-[(3-methyl-1-benzofuran-2-yl)methyl]pyrimidin-4-amine
1-{4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}pyrrolidin-2-one
3-[(3-fluorophenyl)methyl]-N-{[3-(trifluoromethyl)phenyl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[3-(4-chlorobenzoyl)piperidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine
5-(4-benzoylpiperidine-1-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
2-(4-methoxyphenyl)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
1-(3-methyl-3-phenylpiperidin-1-yl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
2-[2-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
N-cyclohexyl-2-methyl-N-(pyridin-2-ylmethyl)imidazo[1,2-a]pyrimidine-3-carboxamide
N-({5-methyl-2-[3-(5-methylthiophene-2-amido)phenyl]-1,3-oxazol-4-yl}methyl)-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)pyrrolidin-3-yl]methanol
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-methyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]benzamide
1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-3-methylpiperidine
1-[(4-fluorophenyl)methyl]-4-(2-methylpyridine-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
1-(3-methoxypropyl)-8-(naphthalen-2-ylmethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-N-(2-hydroxyethyl)-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-4-carboxamide
2,4-dimethyl-N-[4-(4-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
(4aR,7aS)-1-acetyl-4-(1-benzofuran-5-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-ethyl-N-[(5-ethylpyridin-2-yl)methyl]-N,6-dimethylpyrimidin-4-amine
2-amino-4-(4-hydroxy-3,5-dimethoxyphenyl)-6-(propan-2-yl)pyridine-3-carbonitrile
5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
9-[2-(1H-imidazol-1-yl)ethyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
1-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
6-methyl-3-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
4-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[(4-methoxyphenyl)methyl]-1,3-oxazole-4-carboxamide
N-cyclopropyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide