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2-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]pyridin-3-ol
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-oxopropanamide
(4aS,8aR)-1-(2-aminoethyl)-6-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-[(4-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-benzyl-9-[2-(morpholin-2-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,3,5-trimethyl-1H-pyrazole
6-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-methyl-N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidine-3-carbonyl}pyridine
2-(cyclopropylmethyl)-9-(2,4-dimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-1-[1-(2-methoxyphenyl)piperidin-4-yl]-4-propylpyrrolidin-3-yl]acetamide
1-[(2-fluorophenyl)methoxy]-8-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
N-{[7-(cyclohexylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(2-hydroxybutyl)benzamide
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyridin-2-amine
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
2-(5-acetylthiophen-3-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]ethan-1-one
(2R,3S,6R)-5-(1,3-benzothiazole-6-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-1-(furan-2-ylmethyl)piperidine
5-methoxy-4-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,4-dihydropyridine-2-carboxamide
2-{5-[1-(4-tert-butylbenzoyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
2-ethoxy-5-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}pyridine
2-(2,5-dioxoimidazolidin-1-yl)-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}acetamide
2-(5-acetylthiophen-3-yl)-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
(3S,4S)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-{[2-(difluoromethoxy)phenyl]methyl}-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
N-[(3S,4R)-4-(4-methylphenyl)-1-(oxan-4-yl)pyrrolidin-3-yl]acetamide
1-cyclopentyl-5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
9-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-3-oxa-9-azaspiro[5.5]undecane
ethyl 1-[(1-benzylpiperidin-4-yl)methyl]-1H-imidazole-2-carboxylate
(1S,5R)-6-benzyl-3-[(3,4-dimethoxypyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-(1-methylpiperidin-4-yl)-3-[1-(quinolin-2-ylmethyl)piperidin-3-yl]propanamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-6-methylpyridine-3-carboxamide
7-(2,5-dimethoxy-4-methylbenzenesulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{3-[(3-methoxyphenyl)methyl]-1,2-oxazole-5-carbonyl}azocane
4-(3-ethyl-1H-indole-2-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-({[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
(3aR,6aS)-N-{4-[2-(pyridin-2-yl)ethyl]phenyl}-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
4-{1-[1-(2-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]propan-2-yl}morpholine
N-cyclopentyl-2-[2-(dimethylamino)pyrimidin-5-yl]-7-methylquinoline-4-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-methyl-4-[5-methyl-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]piperazine
1-(cyclohex-1-en-1-ylmethyl)-3-(3,5-dimethoxyphenyl)urea
N3-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
2-(dimethylamino)-1-[2-(4-methylpentyl)morpholin-4-yl]ethan-1-one
3-methyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-1H-pyrazole-5-carboxamide
3-({[(2-fluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
({2-[(dimethylamino)methyl]phenyl}methyl)(methyl)[(2-methyl-1H-imidazol-4-yl)methyl]amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide