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1-(pyridin-2-yl)-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(2-oxopiperidin-1-yl)butanamide
6-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2-methoxyethyl)-2-(3-methyl-1,2-oxazol-5-yl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
5-chloro-3-methyl-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-indole-2-carboxamide
(3S,4S)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
2-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
N-{3-oxo-3-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}methanesulfonamide
1-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
4-[(2R)-2-amino-4-methylpentanamido]-N-phenylpiperidine-1-carboxamide
2-{5-[1-(3-hydroxypyridine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
N-[2-(4-hydroxy-1-methylpiperidin-4-yl)ethyl]-4-(trifluoromethyl)benzamide
N-cyclopentyl-1-(2-methylpropyl)-5-(pyrazine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-4-(methoxymethyl)piperidine
ethyl 4-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(methylsulfanyl)pyrimidine-5-carboxylate
N-ethyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-(3-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-3-oxopropyl)pyrrolidin-2-one
4-[(furan-2-ylmethyl)amino]-5-methyl-N-(2-phenylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
2-cyclopentyl-8-(3-fluoropyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]furan-3-carboxamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(2-fluoro-3-methylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
2-(1H-imidazol-4-yl)-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
3-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-3,4-dihydroquinazolin-4-one
1-(4-ethylpiperazin-1-yl)-3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}propan-1-one
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(piperidine-1-carbonyl)piperidine
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]propanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-2-one
5-cyclopropanecarbonyl-1'-(2-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methoxyphenyl)methyl]-N-methylacetamide
[(3R,4R)-1-(4-chloro-3-fluorobenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-3-[2-(4-methylphenoxy)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
N-cyclopropyl-5-[(8-hydroxyquinolin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-(1-benzothiophen-2-ylmethyl)-4-(2-methoxyethyl)piperazine
3-[(dimethylamino)methyl]-1-(5-fluoro-3-methyl-1H-indole-2-carbonyl)pyrrolidin-3-ol
1-[2-(propylsulfanyl)phenyl]-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
2-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]azetidin-3-yl}pyridine
1-cyclopentyl-4-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperazine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N-[3-(furan-2-yl)propyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-{[3-methyl-7-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
7-methoxy-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-amino-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)cyclobutane-1-carboxamide
1'-(2-ethoxyethyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(1S,6R)-N-[(2,4-dichlorophenyl)methyl]-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
1-benzyl-5-acetamido-2-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-1,3-benzodiazole-7-carboxamide
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-cycloheptylpiperidine
1-(3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
2-methoxy-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide