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1-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
N-ethyl-1-[(3-fluorophenyl)methyl]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
8-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-[2-(dimethylamino)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(4-tert-butyl-1,3-thiazol-2-yl)-2-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}acetamide
[3-(prop-2-en-1-yl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidin-3-yl]methanol
methyl (2S)-2-[(2-cyclobutaneamido-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-5-yl)formamido]-2-phenylacetate
5-{2-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]morpholin-4-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-[4-({1-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}methyl)phenyl]acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-3-(pyridin-3-yl)propanamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 2-(azepane-1-sulfonyl)-6-[(2-ethoxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}-4-methylpiperazine
6-tert-butyl-1-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-ethylpropanamide
N2-benzyl-N2,7,7-trimethyl-N5-(pyridin-4-ylmethyl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(thiophen-2-ylmethyl)piperidine-4-carboxamide
4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-1,2,3-triazole
7-methyl-4-{2-[3-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}-2H-chromen-2-one
3-(2-methoxyethyl)-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidine-3-carboxylic acid
methyl (2S,4R)-4-(3-fluorobenzamido)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidine-2-carboxylate
4-chloro-N-(2-methoxyethyl)-1-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-({[1-(thian-4-yl)piperidin-4-yl]carbamoyl}amino)benzamide
N-benzyl-2-[1-cyclopentyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
4-(ethylamino)-N-(3-methoxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-(1-methyl-1H-imidazol-2-yl)-1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
N-butyl-2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
ethyl 1-{[5-(methoxymethyl)furan-2-yl]methyl}-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-(cyclohex-1-en-1-yl)-N-({1-[(2-methylpyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
3-oxo-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
4-{[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
N-{2-[1-benzyl-3-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
6-(aminomethyl)-N-[1-(thiophen-3-yl)propan-2-yl]pyrimidin-4-amine
3-[2-(4-benzylpiperazin-1-yl)-2-oxoethyl]-1-cyclopropyl-3-(2-methylphenyl)pyrrolidine-2,5-dione
5-(3-methoxyphenoxymethyl)-N-(1-propylpiperidin-4-yl)-1,2-oxazole-3-carboxamide
4-(4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-[6-methyl-2-(methylamino)pyrimidin-4-yl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
2-[6-(dimethylamino)pyridine-3-carbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-(2-chloro-5-fluorophenyl)-4-(morpholin-4-yl)piperidine-1-carboxamide
N-({1-[3-(2-oxopyrrolidin-1-yl)benzoyl]piperidin-3-yl}methyl)furan-2-carboxamide
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(2-phenylpropyl)acetamide
N'1-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)cyclopropane-1,1-dicarboxamide
3-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
2-{2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]phenoxy}acetic acid
1-[4-({[2-(2-fluorophenyl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
3-(2-ethylbutyl)-8-(2-methoxybutanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}propanamide